Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 50000842
Affinity DataIC50: 0.00700nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair















