Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50030795
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301551(trans-methyl 4-(3-(2-(4-(trifluoromethoxy)benzylca...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301549(trans-2-(5-(4-chlorophenyl)-4,5-dihydroisoxazol-3-...)
Affinity DataIC50: 430nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301550(trans-2-(5-(3-chlorophenyl)-4,5-dihydroisoxazol-3-...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301548(trans-N-(4-(trifluoromethoxy)benzyl)-2-(5-(4-(trif...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301546(trans-2-(5-phenyl-4,5-dihydrooxazol-2-yl)-N-(4-(tr...)
Affinity DataIC50: 620nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301552(trans-methyl 3-(3-(2-(4-(trifluoromethoxy)benzylca...)
Affinity DataIC50: 710nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301547(trans-2-(5-phenyl-4,5-dihydroisoxazol-3-yl)-N-(4-(...)
Affinity DataIC50: 780nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50178861(trans-N1-methyl-N1-((2'-sulfamoylbiphenyl-4-yl)met...)
Affinity DataIC50: 830nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301553(trans-2-(5-methyl-5-phenyl-4,5-dihydroisoxazol-3-y...)
Affinity DataIC50: 960nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301545(trans-2-(4-(4-chlorophenyl)-4,5-dihydrooxazol-2-yl...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301555(trans-N-(4-isopropoxybenzyl)-2-(5-methyl-5-phenyl-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50301554(trans-2-(5-methyl-5-phenyl-4,5-dihydroisoxazol-3-y...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human Nav1.7 channel expressed in HEK cells by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed