Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 5679
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 22nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92582(ETP-45798, 9)
Affinity DataIC50: 114nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM50328064(CHEMBL1258354 | ETP-7382 | N-(3-methoxyphenyl)-1-m...)
Affinity DataIC50: 400nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92586(ETP-45867, 14)
Affinity DataIC50: 840nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92584(ETP-45874, 11)
Affinity DataIC50: 970nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92583(ETP-45799, 10)
Affinity DataIC50: 1.66E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92588(ETP-45875, 16)
Affinity DataIC50: 3.53E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92574(ETP-5935)
Affinity DataIC50: 4.90E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92579(ETP-45419, 3d)
Affinity DataIC50: 5.51E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92587(ETP-45871, 15)
Affinity DataIC50: 5.80E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92589(ETP-45876, 17)
Affinity DataIC50: 7.00E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM50298309(ETP-7146 | CHEMBL574533 | N-(3-methoxyphenyl)-1-me...)
Affinity DataIC50: 9.20E+3nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92573(ETP-8162)
Affinity DataIC50: 1.26E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92575(ETP-6531)
Affinity DataIC50: 1.26E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 1.31E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92581(ETP-45797, 7)
Affinity DataIC50: 1.61E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 1.68E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92576(ETP-45415, 3a)
Affinity DataIC50: 3.51E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92577(ETP-45416, 3b)
Affinity DataIC50: 3.68E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 3.98E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92578(ETP-45654, 3c)
Affinity DataIC50: 5.00E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92580(ETP-45700, 6)
Affinity DataIC50: 5.00E+4nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 1.29E+5nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 1.52E+5nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Spanish National Cancer Research Center (Cnio)

LigandPNGBDBM92585(ETP-45658, 13)
Affinity DataIC50: 7.17E+5nMAssay Description:Kinase assay using PI3K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed