Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50030512
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataEC50:  0.390nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297345((5S,8S,13R,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297343((5S,8S,13S,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297345((5S,8S,13R,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  1.85nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297345((5S,8S,13R,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  2.33nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataKi:  2.46nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50010704(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  6.18nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297345((5S,8S,13R,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataKi:  10.9nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297343((5S,8S,13S,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  87.2nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297343((5S,8S,13S,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  763nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347(CHEMBL564095 | (2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50297343((5S,8S,13S,Z)-13-((S)-2-amino-3-(4-hydroxyphenyl)p...)
Affinity DataKi:  7.67E+3nMAssay Description:Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed