Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50030944
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 1.07nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304334(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-tropane | ...)
Affinity DataIC50: 10.2nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 11.5nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304334(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-tropane | ...)
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]granisectron from 5HT3 receptor in Wistar rat forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]granisectron from 5HT3 receptor in Wistar rat forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304333(3alpha-(2'-Indolecarbonyloxy)-nortropane | CHEMBL5...)
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]granisectron from 5HT3 receptor in Wistar rat forebrainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415201(CHEMBL611364)
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415204(CHEMBL596443)
Affinity DataIC50: 41.7nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415205(CHEMBL595797)
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415208(CHEMBL608418)
Affinity DataIC50: 58.9nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415210(CHEMBL608417)
Affinity DataIC50: 60.3nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 70.8nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415211(CHEMBL595791)
Affinity DataIC50: 72.4nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415206(CHEMBL596257)
Affinity DataIC50: 79.4nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415203(CHEMBL595116)
Affinity DataIC50: 89.1nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415209(CHEMBL596237)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415202(CHEMBL611365)
Affinity DataIC50: 129nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415200(CHEMBL610170)
Affinity DataIC50: 166nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304333(3alpha-(2'-Indolecarbonyloxy)-nortropane | CHEMBL5...)
Affinity DataIC50: 234nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304334(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-tropane | ...)
Affinity DataIC50: 1.58E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415211(CHEMBL595791)
Affinity DataIC50: 1.91E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415203(CHEMBL595116)
Affinity DataIC50: 1.91E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304334(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-tropane | ...)
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415208(CHEMBL608418)
Affinity DataIC50: 4.27E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415203(CHEMBL595116)
Affinity DataIC50: 4.27E+3nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415210(CHEMBL608417)
Affinity DataIC50: 4.68E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415211(CHEMBL595791)
Affinity DataIC50: 5.50E+3nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415205(CHEMBL595797)
Affinity DataIC50: 5.62E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415207(CHEMBL594193)
Affinity DataIC50: 7.59E+3nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415210(CHEMBL608417)
Affinity DataIC50: 7.94E+3nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415205(CHEMBL595797)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415201(CHEMBL611364)
Affinity DataIC50: 1.12E+4nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415201(CHEMBL611364)
Affinity DataIC50: 2.09E+4nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50415208(CHEMBL608418)
Affinity DataIC50: 2.29E+4nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed