Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50035894
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 70nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010733(CHEMBL540546 | 5-[2-(Ethyl-phenethyl-amino)-ethyl]...)
Affinity DataIC50: 230nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010731(CHEMBL543838 | 2-Fluoro-5-[2-(phenethyl-propyl-ami...)
Affinity DataIC50: 250nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010729(CHEMBL538012 | 2-Fluoro-4-[2-(phenethyl-propyl-ami...)
Affinity DataIC50: 580nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010732(CHEMBL541304 | 5-(2-Dipropylamino-ethyl)-2-fluoro-...)
Affinity DataIC50: 950nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010734(CHEMBL540036 | 5-[2-(Ethyl-propyl-amino)-ethyl]-2-...)
Affinity DataIC50: 1.97E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010730(CHEMBL545240 | 5-(2-Amino-ethyl)-2-fluoro-phenol; ...)
Affinity DataIC50: 4.64E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]spiperone binding to dopamine receptor D2 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010730(CHEMBL545240 | 5-(2-Amino-ethyl)-2-fluoro-phenol; ...)
Affinity DataIC50: 6.15E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010733(CHEMBL540546 | 5-[2-(Ethyl-phenethyl-amino)-ethyl]...)
Affinity DataIC50: 8.00E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010731(CHEMBL543838 | 2-Fluoro-5-[2-(phenethyl-propyl-ami...)
Affinity DataIC50: 1.09E+4nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010734(CHEMBL540036 | 5-[2-(Ethyl-propyl-amino)-ethyl]-2-...)
Affinity DataIC50: 1.11E+4nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010732(CHEMBL541304 | 5-(2-Dipropylamino-ethyl)-2-fluoro-...)
Affinity DataIC50: 1.14E+4nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50010729(CHEMBL538012 | 2-Fluoro-4-[2-(phenethyl-propyl-ami...)
Affinity DataIC50: 3.80E+4nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed