Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50030963
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304572(5-Oxo-5,6-dihydro-pyrido[2',1':2,3]imidazo[4,5-c]i...)
Affinity DataIC50: 36nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304575(10-Methyl-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoqui...)
Affinity DataIC50: 470nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304570(10-Methyl-pyrimido[1',2':1,2]imidazo[5,4-c]isoquin...)
Affinity DataIC50: 560nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304573(Pyrido[2',1':2,3]imidazo[4,5-c]isoquinolin-5-(6H)-...)
Affinity DataIC50: 850nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304567(6H-Pyrimido[4',3':1,2]imidazo[5,4-c]isoquinolin-5-...)
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304574(11-Methyl-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoqui...)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304569(6H-Naphto[2',1':1,2]imidazo[5,4-c]isoquinolin-5-on...)
Affinity DataIC50: 4.11E+3nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304576(9-Methyl-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoquin...)
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304568(6H-Pyrimido[1',2':1,2]imidazo[5,4-c]isoquinolin-5-...)
Affinity DataIC50: 5.78E+3nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304565(10-Chloro-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoqui...)
Affinity DataIC50: 5.87E+3nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM27502(CHEMBL127336 | 3,4-dihydro-5-(4-(1-piperidinyl)but...)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304579(9-Bromo-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoquino...)
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304578(9-Chloro-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoquin...)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304566(8,10-Dimethyl-6H-pyrido[2',1':1,2]imidazo[5,4-c]is...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304571(10-Methoxy-6H-pyrimido[3',4':1,2]imidazo[5,4-c]iso...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Sookmyung Women'S University

Curated by ChEMBL
LigandPNGBDBM50304577(8-Methyl-6H-pyrido[2',1':1,2]imidazo[5,4-c]isoquin...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed