Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50030653
TargetBaculoviral IAP repeat-containing protein 5(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM26673(CHEMBL391586 | 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4...)
Affinity DataKd:  5.70E+3nMAssay Description:Inhibition of survivinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50209209(6-(5-bromo-2-hydroxyphenyl)-4-(2,5-dichlorophenyl)...)
Affinity DataKd:  800nMAssay Description:Inhibition of survivinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM26673(CHEMBL391586 | 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4...)
Affinity DataIC50: 50nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50299695(4-(4-Ethoxyphenyl)-2-imino-6-(thiophen-3-yl)-1,2-d...)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human recombinant PDE3A by fluorescence polarization assay using cAMP as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50299695(4-(4-Ethoxyphenyl)-2-imino-6-(thiophen-3-yl)-1,2-d...)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human recombinant PDE3A by fluorescence polarization assay using cGMP as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed