Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50031348
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM27641(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-[(...)
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311688(N-(2-methoxybenzyl)-1-(3-((2-(methylamino)ethylami...)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311707(1-(3-((2-(methylamino)ethylamino)methyl)phenyl)-N-...)
Affinity DataIC50: 320nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311700(N-(5-fluoro-2-methoxybenzyl)-1-(3-((2-(methylamino...)
Affinity DataIC50: 710nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311699(N-((2,3-dihydrobenzo[b][1,4]dioxin-5-yl)methyl)-1-...)
Affinity DataIC50: 710nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311698(N-(2-ethoxybenzyl)-1-(3-((2-(methylamino)ethylamin...)
Affinity DataIC50: 900nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311689(1-(3-((2-aminoethylamino)methyl)phenyl)-N-(2-metho...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311697(N-(2-ethylbenzyl)-1-(3-((2-(methylamino)ethylamino...)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311706(N-(2-(1H-indol-3-yl)ethyl)-1-(3-((2-(methylamino)e...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311708(N-((2-methoxynaphthalen-1-yl)methyl)-1-(3-((2-(met...)
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311703(N-(cyclohexylmethyl)-1-(3-((2-(methylamino)ethylam...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311705(N-((1H-benzo[d]imidazol-2-yl)methyl)-1-(3-((2-(met...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311684((S)-1-(3-((2-aminopropanethioamido)methyl)phenyl)-...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311704(N-((1-methyl-1H-benzo[d]imidazol-2-yl)methyl)-1-(3...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311709(1-(4-fluoro-3-((2-(methylamino)ethylamino)methyl)p...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311701(1-(3-((2-(methylamino)ethylamino)methyl)phenyl)-N-...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311691(1-(3-((2-(ethylamino)ethylamino)methyl)phenyl)-N-(...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311690(1-(3-((2-(dimethylamino)ethylamino)methyl)phenyl)-...)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311710(N-(2-methoxybenzyl)-1-(4-methyl-3-((2-(methylamino...)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311702(N-(2-aminobenzyl)-1-(3-((2-(methylamino)ethylamino...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311712(5-(2-methoxybenzyl)-8-((2-(methylamino)ethylamino)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311695(N-benzyl-1-(3-((2-(methylamino)ethylamino)methyl)p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311696(1-(3-((2-(methylamino)ethylamino)methyl)phenyl)-N-...)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311687((S)-1-(3-(5-(1-aminoethyl)-1,2,4-oxadiazol-3-yl)ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311686((S)-1-(3-(5-(1-aminoethyl)-1H-1,2,4-triazol-3-yl)p...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311685((S)-1-(3-((2-hydroxypropanamido)methyl)phenyl)-N-(...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311692(N-(2-methoxybenzyl)-1-(3-((pyrrolidin-3-ylamino)me...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311711(N-(2-methoxybenzyl)-1-(3-((2-(methylamino)ethylami...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311694(N-(2-methoxybenzyl)-1-(3-(2-(methylamino)ethylcarb...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311683((S)-1-(3-(2-(2-aminopropanamido)ethyl)phenyl)-N-(2...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Mouse)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311693(N-(2-methoxybenzyl)-1-(3-(1-(2-(methylamino)ethyla...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of N-terminal His-tagged mouse recombinant CARM1 expressed in Sf9 cells by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETD7(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50311688(N-(2-methoxybenzyl)-1-(3-((2-(methylamino)ethylami...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human recombinant SET7/9 expressed in Escherichia coli by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50311688(N-(2-methoxybenzyl)-1-(3-((2-(methylamino)ethylami...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal GST-tagged human recombinant PRMT1 expressed in Escherichia coli by microbeta countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed