Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50030669
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299871(5-(1-ethyl-1-hydroxy-3,3-dimethyl-2,3-dihydro-1H-i...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299872(5-(3,3-dimethyl-1-oxo-2,3-dihydro-1H-inden-5-yl)-1...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299873(5-(1-hydroxy-3,3-dimethyl-2,3-dihydro-1H-inden-5-y...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299874(1-methyl-5-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1H-py...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299875(5-(1-(hydroxyimino)-2,3-dihydro-1H-inden-5-yl)-1-m...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299876(5-(1-(hydroxyimino)-3-methyl-2,3-dihydro-1H-inden-...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299877(5-(1-(hydroxyimino)-3,3-dimethyl-2,3-dihydro-1H-in...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299878(5-(1-hydroxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-1...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299879(5-(1-hydroxy-3-methyl-2,3-dihydro-1H-inden-5-yl)-1...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299880(5-(1-hydroxy-3,3-dimethyl-1-(prop-2-ynyl)-2,3-dihy...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299870(5-(1-hydroxy-1,3,3-trimethyl-2,3-dihydro-1H-inden-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299880(5-(1-hydroxy-3,3-dimethyl-1-(prop-2-ynyl)-2,3-dihy...)
Affinity DataIC50: 3nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299878(5-(1-hydroxy-2,3-dihydro-1H-inden-5-yl)-1-methyl-1...)
Affinity DataIC50: 10nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299877(5-(1-(hydroxyimino)-3,3-dimethyl-2,3-dihydro-1H-in...)
Affinity DataIC50: 14nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299879(5-(1-hydroxy-3-methyl-2,3-dihydro-1H-inden-5-yl)-1...)
Affinity DataIC50: 18nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299874(1-methyl-5-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1H-py...)
Affinity DataIC50: 34nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299876(5-(1-(hydroxyimino)-3-methyl-2,3-dihydro-1H-inden-...)
Affinity DataIC50: 65nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299881(5-(3-chlorophenyl)-3,3-dimethyl-2,3-dihydro-1H-ind...)
Affinity DataIC50: 66nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299882(5-(3,4-dichlorophenyl)-3,3-dimethyl-2,3-dihydro-1H...)
Affinity DataIC50: 79nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299875(5-(1-(hydroxyimino)-2,3-dihydro-1H-inden-5-yl)-1-m...)
Affinity DataIC50: 132nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299883(3-(3,3-dimethyl-1-oxo-2,3-dihydro-1H-inden-5-yl)be...)
Affinity DataIC50: 195nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299884(3,3-dimethyl-5-m-tolyl-2,3-dihydro-1H-inden-1-one ...)
Affinity DataIC50: 225nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299885(3,3-dimethyl-5-m-tolyl-2,3-dihydro-1H-inden-1-one ...)
Affinity DataIC50: 316nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299886(3-(1-(hydroxyimino)-3,3-dimethyl-2,3-dihydro-1H-in...)
Affinity DataIC50: 317nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299887(5-(3,4-dichlorophenyl)-3,3-dimethyl-2,3-dihydro-1H...)
Affinity DataIC50: 456nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50299888(5-(3-chlorophenyl)-3,3-dimethyl-2,3-dihydro-1H-ind...)
Affinity DataIC50: 490nMAssay Description:Inhibition of progesterone receptor in human T47D cells assessed as progesteron-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed