Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50004266
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50129793(N-methyl-[11C]2-(40-methylaminophenyl)-6-hydroxy b...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480917(CHEMBL566354)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480918(CHEMBL578982)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479543(CHEMBL510384)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480919(CHEMBL568061)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed