Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50038997
TargetLipoxygenase(Potato)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303170(N-Acetyl-5-(N-difluoromethyl-1,2-dihydropyrid-2-on...)
Affinity DataIC50: 280nMAssay Description:Inhibition of potato 5-LOX after 5 mins by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetLipoxygenase(Potato)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303169(N-Acetyl-4-(N-difluoromethyl-1,2-dihydropyrid-2-on...)
Affinity DataIC50: 320nMAssay Description:Inhibition of potato 5-LOX after 5 mins by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Bovine)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoic acid | 2-(acetyloxy)benzoate ...)
Affinity DataIC50: 350nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetLipoxygenase(Potato)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303172(5-(N-Difluoromethyl-1,2-dihydropyrid-2-one-4-yl)sa...)
Affinity DataIC50: 370nMAssay Description:Inhibition of potato 5-LOX after 5 mins by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303172(5-(N-Difluoromethyl-1,2-dihydropyrid-2-one-4-yl)sa...)
Affinity DataIC50: 980nMAssay Description:Inhibition of human recombinant COX-2 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50009859((RS)-ibuprofen | CHEMBL521 | 2-(4-isobutylphenyl)p...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant COX-2 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoic acid | 2-(acetyloxy)benzoate ...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant COX-2 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303170(N-Acetyl-5-(N-difluoromethyl-1,2-dihydropyrid-2-on...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant COX-2 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Bovine)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50009859((RS)-ibuprofen | CHEMBL521 | 2-(4-isobutylphenyl)p...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLipoxygenase(Potato)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM4375(3,4-Dihydroxycinnamate, XVII | cid_689043 | Caffei...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of potato 5-LOX after 5 mins by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303171(4-(N-Difluoromethyl-1,2-dihydropyrid-2-one-4-yl)sa...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human recombinant COX-2 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetLipoxygenase(Potato)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303171(4-(N-Difluoromethyl-1,2-dihydropyrid-2-one-4-yl)sa...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of potato 5-LOX after 5 mins by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Bovine)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303172(5-(N-Difluoromethyl-1,2-dihydropyrid-2-one-4-yl)sa...)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303169(N-Acetyl-4-(N-difluoromethyl-1,2-dihydropyrid-2-on...)
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of human recombinant COX-2 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Bovine)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303170(N-Acetyl-5-(N-difluoromethyl-1,2-dihydropyrid-2-on...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Bovine)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303169(N-Acetyl-4-(N-difluoromethyl-1,2-dihydropyrid-2-on...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Bovine)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50303171(4-(N-Difluoromethyl-1,2-dihydropyrid-2-one-4-yl)sa...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed