Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50030992
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304919(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304926(N-(3,4-dimethyl-5-(piperidin-1-ylsulfonyl)phenyl)-...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304916(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-3,3,...)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304925(N-(3,4-dimethyl-5-(thiazolidin-3-ylsulfonyl)phenyl...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304935(N-[3-(1,1-Dioxo-1lambda*6*-thiomorpholine-4-sulfon...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304924(N-(3-(azepan-1-ylsulfonyl)-4,5-dimethylphenyl)-2,2...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304918(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304916(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-3,3,...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304920(2,2-dimethyl-N-(7-(morpholinosulfonyl)-2,3-dihydro...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304925(N-(3,4-dimethyl-5-(thiazolidin-3-ylsulfonyl)phenyl...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304926(N-(3,4-dimethyl-5-(piperidin-1-ylsulfonyl)phenyl)-...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304921(2,2-dimethyl-N-(4-(morpholinosulfonyl)-5,6,7,8-tet...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304914(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2,...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304917(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304935(N-[3-(1,1-Dioxo-1lambda*6*-thiomorpholine-4-sulfon...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304918(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304924(N-(3-(azepan-1-ylsulfonyl)-4,5-dimethylphenyl)-2,2...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304917(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataEC50:  38nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304915(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)pival...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304934((R)-N-(3-(2-(hydroxymethyl)pyrrolidin-1-ylsulfonyl...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304923(N-(3-(N-(cyclopropylmethyl)sulfamoyl)-4,5-dimethyl...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304914(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2,...)
Affinity DataEC50:  66nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304933((S)-N-(3-(3-hydroxypyrrolidin-1-ylsulfonyl)-4,5-di...)
Affinity DataEC50:  73nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304919(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataEC50:  82nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304933((S)-N-(3-(3-hydroxypyrrolidin-1-ylsulfonyl)-4,5-di...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304915(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)pival...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304922(N-(3-(N-cyclopentylsulfamoyl)-4,5-dimethylphenyl)-...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304922(N-(3-(N-cyclopentylsulfamoyl)-4,5-dimethylphenyl)-...)
Affinity DataEC50:  98nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304934((R)-N-(3-(2-(hydroxymethyl)pyrrolidin-1-ylsulfonyl...)
Affinity DataEC50:  98nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304929(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-4-me...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304927(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2-me...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304923(N-(3-(N-(cyclopropylmethyl)sulfamoyl)-4,5-dimethyl...)
Affinity DataEC50:  135nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304919(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304930(2,2-dimethyl-N-(4-methyl-3-(morpholinosulfonyl)phe...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304932(2,2-dimethyl-N-(2,3,4-trimethyl-5-(morpholinosulfo...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304926(N-(3,4-dimethyl-5-(piperidin-1-ylsulfonyl)phenyl)-...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304931(N-(2,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  760nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304916(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-3,3,...)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304918(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  830nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304914(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2,...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304921(2,2-dimethyl-N-(4-(morpholinosulfonyl)-5,6,7,8-tet...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304921(2,2-dimethyl-N-(4-(morpholinosulfonyl)-5,6,7,8-tet...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304920(2,2-dimethyl-N-(7-(morpholinosulfonyl)-2,3-dihydro...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304920(2,2-dimethyl-N-(7-(morpholinosulfonyl)-2,3-dihydro...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304924(N-(3-(azepan-1-ylsulfonyl)-4,5-dimethylphenyl)-2,2...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304928(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2-hy...)
Affinity DataKi:  2.08E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304925(N-(3,4-dimethyl-5-(thiazolidin-3-ylsulfonyl)phenyl...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Adolor

Curated by ChEMBL
LigandPNGBDBM50304917(N-(3,4-dimethyl-5-(morpholinosulfonyl)phenyl)-2,2-...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
Displayed 1 to 50 (of 54 total ) | Next | Last >>
Jump to: