Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 50030995
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304978((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-chloroben...)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304987((S)-4-((2-bromobenzyl)(1-propionylpyrrolidin-3-yl)...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304972((S)-2-chloro-4-((2-chlorobenzyl)(1-(methylsulfonyl...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304957((S)-2-chloro-4-((2-methylbenzyl)(1-propionylpyrrol...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304961(2-chloro-4-(((S)-1-((S)-2-hydroxypropanoyl)pyrroli...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304973((S)-4-((2-bromobenzyl)(1-(methylsulfonyl)pyrrolidi...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304977((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-methylben...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304973((S)-4-((2-bromobenzyl)(1-(methylsulfonyl)pyrrolidi...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304972((S)-2-chloro-4-((2-chlorobenzyl)(1-(methylsulfonyl...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304987((S)-4-((2-bromobenzyl)(1-propionylpyrrolidin-3-yl)...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304978((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-chloroben...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304975((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-(trifluor...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50298028(2-chloro-4-{[(3S)-1-methylpyrrolidin-3-yl][2-(trif...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304968((S)-2-chloro-4-((1-(isobutylsulfonyl)pyrrolidin-3-...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304964((S)-2-chloro-4-((1-(methylsulfonyl)pyrrolidin-3-yl...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304976((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-fluoroben...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304977((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-methylben...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304975((S)-methyl 3-((3-chloro-4-cyanophenyl)(2-(trifluor...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304964((S)-2-chloro-4-((1-(methylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50: 13nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50298028(2-chloro-4-{[(3S)-1-methylpyrrolidin-3-yl][2-(trif...)
Affinity DataIC50: 16nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304974(2-chloro-4-{(2-methylbenzyl)[(3S)-1-(methylsulfony...)
Affinity DataIC50: 16nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304957((S)-2-chloro-4-((2-methylbenzyl)(1-propionylpyrrol...)
Affinity DataIC50: 16nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304980((S)-methyl 3-((3-chloro-4-cyanophenyl)(5-fluoro-2-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304979((S)-methyl 3-((3-chloro-4-cyanophenyl)(2,3-difluor...)
Affinity DataIC50: 20nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304971((S)-2-chloro-4-((2-fluorobenzyl)(1-(methylsulfonyl...)
Affinity DataIC50: 20nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304984((S)-2-chloro-4-((1-propionylpyrrolidin-3-yl)(2-(tr...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304985((S)-2-chloro-4-((1-isobutyrylpyrrolidin-3-yl)(2-(t...)
Affinity DataIC50: 25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304984((S)-2-chloro-4-((1-propionylpyrrolidin-3-yl)(2-(tr...)
Affinity DataIC50: 25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304959((S)-2-chloro-4-((2,5-dichlorobenzyl)(1-propionylpy...)
Affinity DataIC50: 25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304974(2-chloro-4-{(2-methylbenzyl)[(3S)-1-(methylsulfony...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304958((S)-2-chloro-4-((5-fluoro-2-methylbenzyl)(1-propio...)
Affinity DataIC50: 25nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304981((S)-ethyl 3-((3-chloro-4-cyanophenyl)(5-fluoro-2-m...)
Affinity DataIC50: 30nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304983((S)-4-((1-acetylpyrrolidin-3-yl)(2-(trifluoromethy...)
Affinity DataIC50: 30nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304961(2-chloro-4-(((S)-1-((S)-2-hydroxypropanoyl)pyrroli...)
Affinity DataIC50: 32nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304983((S)-4-((1-acetylpyrrolidin-3-yl)(2-(trifluoromethy...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304971((S)-2-chloro-4-((2-fluorobenzyl)(1-(methylsulfonyl...)
Affinity DataEC50:  36nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304965((S)-2-chloro-4-((1-(ethylsulfonyl)pyrrolidin-3-yl)...)
Affinity DataIC50: 40nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304966((S)-2-chloro-4-((1-(isopropylsulfonyl)pyrrolidin-3...)
Affinity DataIC50: 40nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304980((S)-methyl 3-((3-chloro-4-cyanophenyl)(5-fluoro-2-...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304986((S)-2-chloro-4-((1-pivaloylpyrrolidin-3-yl)(2-(tri...)
Affinity DataIC50: 50nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304963(2-chloro-4-((2,5-dichlorobenzyl)((S)-1-((S)-2-hydr...)
Affinity DataIC50: 50nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304982((S)-isopropyl 3-((3-chloro-4-cyanophenyl)(5-fluoro...)
Affinity DataIC50: 50nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304990((S)-4-((1-(butylsulfonyl)pyrrolidin-3-yl)(2-(trifl...)
Affinity DataIC50: 63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304969((S)-4-(benzyl(1-(methylsulfonyl)pyrrolidin-3-yl)am...)
Affinity DataIC50: 63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304988((S)-methyl 3-(benzyl(3-chloro-4-cyanophenyl)amino)...)
Affinity DataIC50: 63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304960(2-chloro-4-(((S)-1-((S)-2-hydroxypropanoyl)pyrroli...)
Affinity DataIC50: 63nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304958((S)-2-chloro-4-((5-fluoro-2-methylbenzyl)(1-propio...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at PR in human T47D cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304962(2-chloro-4-((5-fluoro-2-methylbenzyl)((S)-1-((S)-2...)
Affinity DataIC50: 79nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304967((S)-2-chloro-4-((1-(propylsulfonyl)pyrrolidin-3-yl...)
Affinity DataIC50: 80nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50304968((S)-2-chloro-4-((1-(isobutylsulfonyl)pyrrolidin-3-...)
Affinity DataIC50: 80nMAssay Description:Inhibition of PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
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