Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50030686
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50300129(CHEMBL572528 | Cibacron Blue 3Ga | CIBACRON BLUE)
Affinity DataIC50: 200nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50300128(4-(BENZHYDRYLOXY)-1-[3-(1H-TETRAAZOL-5-YL)PROPYL]P...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50300127(phenyl(thiophen-2-yl)methanone | NSC-4502 | CHEMBL...)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50300126(Sulfobromophthalein | CHEMBL574431)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50300125(NSC-151248 | (4-methoxyphenyl)(thiophen-2-yl)metha...)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50186231([2,3-dichloro-4-(2-methylidenebutanoyl)phenoxy]ace...)
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetHematopoietic prostaglandin D synthase(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50300124(methyl [5-(phenylsulfinyl)-1H-benzimidazol-2-yl]ca...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 assessed as rate of glutathione-chloro-dinitro benzene conjugationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed