Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50031013
LigandPNGBDBM50305294(5-(6-morpholino-9H-purin-2-yl)pyridin-3-ol | CHEMB...)
Affinity DataIC50: 11nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305295(5-(6-morpholino-9-(piperidin-4-yl)-9H-purin-2-yl)p...)
Affinity DataIC50: 14nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305293((3-(9-(1-(4-(3-(dimethylamino)propoxy)benzyl)piper...)
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305296(5-(9-(1-(4-chlorobenzyl)piperidin-4-yl)-6-morpholi...)
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305291((3-(6-morpholino-9-(1-(4-(pyridin-4-yl)benzyl)pipe...)
Affinity DataIC50: 23nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305304(3-(9-(1-((5-chloropyridin-3-yl)methyl)piperidin-4-...)
Affinity DataIC50: 37nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305303(3-(6-morpholino-9-(1-((6-morpholinopyridin-3-yl)me...)
Affinity DataIC50: 40nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305289((3-(9-(1-(2-fluorobenzyl)piperidin-4-yl)-6-morphol...)
Affinity DataIC50: 42nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305297(5-(9-(1-(4-methylbenzyl)piperidin-4-yl)-6-morpholi...)
Affinity DataIC50: 42nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305292((3-(9-(1-(2,4-difluorophenyl)piperidin-4-yl)-6-mor...)
Affinity DataIC50: 44nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305295(5-(6-morpholino-9-(piperidin-4-yl)-9H-purin-2-yl)p...)
Affinity DataIC50: 44nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305294(5-(6-morpholino-9H-purin-2-yl)pyridin-3-ol | CHEMB...)
Affinity DataIC50: 47nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305305(3-(9-(1-((6-methoxypyridin-3-yl)methyl)piperidin-4...)
Affinity DataIC50: 51nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305305(3-(9-(1-((6-methoxypyridin-3-yl)methyl)piperidin-4...)
Affinity DataIC50: 55nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305307((3-(6-morpholino-9-(piperidin-4-yl)-9H-purin-2-yl)...)
Affinity DataIC50: 57nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305298(5-(9-(1-((6-fluoropyridin-3-yl)methyl)piperidin-4-...)
Affinity DataIC50: 61nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305306((3-(9-(1-benzylpiperidin-4-yl)-6-morpholino-9H-pur...)
Affinity DataIC50: 63nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305300(3-(6-morpholino-9-(piperidin-4-yl)-9H-purin-2-yl)p...)
Affinity DataIC50: 64nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305288((3-(6-morpholino-9-(1-(pyridin-2-ylmethyl)piperidi...)
Affinity DataIC50: 65nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305302(3-(6-morpholino-9-(1-(pyridin-3-ylmethyl)piperidin...)
Affinity DataIC50: 66nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305290((3-(9-(1-(4-fluorobenzyl)piperidin-4-yl)-6-morphol...)
Affinity DataIC50: 70nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305301(3-(9-(1-benzylpiperidin-4-yl)-6-morpholino-9H-puri...)
Affinity DataIC50: 75nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305298(5-(9-(1-((6-fluoropyridin-3-yl)methyl)piperidin-4-...)
Affinity DataIC50: 94nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305296(5-(9-(1-(4-chlorobenzyl)piperidin-4-yl)-6-morpholi...)
Affinity DataIC50: 119nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305300(3-(6-morpholino-9-(piperidin-4-yl)-9H-purin-2-yl)p...)
Affinity DataIC50: 133nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305301(3-(9-(1-benzylpiperidin-4-yl)-6-morpholino-9H-puri...)
Affinity DataIC50: 140nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305299(3-(6-morpholino-9H-purin-2-yl)phenol | CHEMBL59351...)
Affinity DataIC50: 150nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305303(3-(6-morpholino-9-(1-((6-morpholinopyridin-3-yl)me...)
Affinity DataIC50: 152nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305296(5-(9-(1-(4-chlorobenzyl)piperidin-4-yl)-6-morpholi...)
Affinity DataIC50: 160nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305289((3-(9-(1-(2-fluorobenzyl)piperidin-4-yl)-6-morphol...)
Affinity DataIC50: 160nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305302(3-(6-morpholino-9-(1-(pyridin-3-ylmethyl)piperidin...)
Affinity DataIC50: 170nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305287(1-(4-(2-(3-(hydroxymethyl)phenyl)-6-morpholino-9H-...)
Affinity DataIC50: 189nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305304(3-(9-(1-((5-chloropyridin-3-yl)methyl)piperidin-4-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305297(5-(9-(1-(4-methylbenzyl)piperidin-4-yl)-6-morpholi...)
Affinity DataIC50: 204nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305291((3-(6-morpholino-9-(1-(4-(pyridin-4-yl)benzyl)pipe...)
Affinity DataIC50: 223nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305293((3-(9-(1-(4-(3-(dimethylamino)propoxy)benzyl)piper...)
Affinity DataIC50: 265nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305293((3-(9-(1-(4-(3-(dimethylamino)propoxy)benzyl)piper...)
Affinity DataIC50: 300nMAssay Description:Inhibition of PI3Kalpha in human MDA-MB-361 cells assessed as reduction of phosphorylated Akt (T308) level after 4 hrs by Western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305305(3-(9-(1-((6-methoxypyridin-3-yl)methyl)piperidin-4...)
Affinity DataIC50: 306nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305288((3-(6-morpholino-9-(1-(pyridin-2-ylmethyl)piperidi...)
Affinity DataIC50: 310nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305304(3-(9-(1-((5-chloropyridin-3-yl)methyl)piperidin-4-...)
Affinity DataIC50: 341nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305303(3-(6-morpholino-9-(1-((6-morpholinopyridin-3-yl)me...)
Affinity DataIC50: 368nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305298(5-(9-(1-((6-fluoropyridin-3-yl)methyl)piperidin-4-...)
Affinity DataIC50: 570nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305302(3-(6-morpholino-9-(1-(pyridin-3-ylmethyl)piperidin...)
Affinity DataIC50: 583nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305297(5-(9-(1-(4-methylbenzyl)piperidin-4-yl)-6-morpholi...)
Affinity DataIC50: 590nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305290((3-(9-(1-(4-fluorobenzyl)piperidin-4-yl)-6-morphol...)
Affinity DataIC50: 594nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305294(5-(6-morpholino-9H-purin-2-yl)pyridin-3-ol | CHEMB...)
Affinity DataIC50: 620nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305292((3-(9-(1-(2,4-difluorophenyl)piperidin-4-yl)-6-mor...)
Affinity DataIC50: 640nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305307((3-(6-morpholino-9-(piperidin-4-yl)-9H-purin-2-yl)...)
Affinity DataIC50: 683nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50305291((3-(6-morpholino-9-(1-(4-(pyridin-4-yl)benzyl)pipe...)
Affinity DataIC50: 720nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50305288((3-(6-morpholino-9-(1-(pyridin-2-ylmethyl)piperidi...)
Affinity DataIC50: 776nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
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