Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50031275
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310309(N-(3,4-dihydroxyphenylsulfonyl)-N-hexyl-3,4-dihydr...)
Affinity DataIC50: 284nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310311(N-cyclohexyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-d...)
Affinity DataIC50: 594nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310308(N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxy-N-pr...)
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310310(N-benzyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihyd...)
Affinity DataIC50: 4.82E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310301(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3,4-dihydroxyben...)
Affinity DataIC50: 9.32E+3nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310307(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3,5-difluoro-4-h...)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310306(N,N'-(ethane-1,2-diyl)bis(N-ethylbenzenesulfonamid...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310313(N,N'-(ethane-1,2-diyl)bis(N-ethyl-2,5-dihydroxyben...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310305(N,N'-(ethane-1,2-diyl)bis(N-ethyl-4-hydroxybenzene...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310310(N-benzyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihyd...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310312(N,N'-bis(3,4-dihydroxybenzenesulfonyl)piperazine |...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310311(N-cyclohexyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-d...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310312(N,N'-bis(3,4-dihydroxybenzenesulfonyl)piperazine |...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310299(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3,4-dimethoxyben...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310306(N,N'-(ethane-1,2-diyl)bis(N-ethylbenzenesulfonamid...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310305(N,N'-(ethane-1,2-diyl)bis(N-ethyl-4-hydroxybenzene...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310313(N,N'-(ethane-1,2-diyl)bis(N-ethyl-2,5-dihydroxyben...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310309(N-(3,4-dihydroxyphenylsulfonyl)-N-hexyl-3,4-dihydr...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310299(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3,4-dimethoxyben...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310304(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3-hydroxybenzene...)
Affinity DataIC50: 3.43E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310300(N,N'-(ethane-1,2-diyl)bis(3,4-dihydroxybenzenesulf...)
Affinity DataIC50: 5.18E+5nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310307(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3,5-difluoro-4-h...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310308(N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxy-N-pr...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310304(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3-hydroxybenzene...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310303(N,N'-(hexane-1,6-diyl)bis(3,4-dihydroxybenzenesulf...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310302(N,N'-(butane-1,4-diyl)bis(3,4-dihydroxybenzenesulf...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310303(N,N'-(hexane-1,6-diyl)bis(3,4-dihydroxybenzenesulf...)
Affinity DataIC50: 1.38E+6nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310300(N,N'-(ethane-1,2-diyl)bis(3,4-dihydroxybenzenesulf...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetAntithrombin-III(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310301(N,N'-(ethane-1,2-diyl)bis(N-ethyl-3,4-dihydroxyben...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of antithrombin-3 assessed as residual alpha-thrombin activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Eastern Michigan University

Curated by ChEMBL
LigandPNGBDBM50310302(N,N'-(butane-1,4-diyl)bis(3,4-dihydroxybenzenesulf...)
Affinity DataIC50: 3.00E+6nMAssay Description:Inhibition of human recombinant PAI1 assessed as rate of AMC release after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed