Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50039015
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303986(Ethyl 2-Methyl-3-(4-(2-(4-methyl-2-propyl-1H-benzo...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at PPARalpha assessed as receptor transactivation by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at PPARalpha assessed as receptor transactivation by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303975(3'-(4-(2-(1H-Tetrazol-5-yl)ethyl)benzyl)-1,7'-dime...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303976(3'-(2-(4-(2-(1H-Tetrazol-5-yl)ethyl)phenoxy)ethyl)...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303977(3-(4-(2-(1,7'-Dimethyl-2'-propyl-1H,3'H-2,5'-biben...)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303979(Ethyl 3-(4-(2-(1,7'-Dimethyl-2'-propyl-1H,3'H-2,5'...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303978(1-(4-(2-(1H-tetrazol-5-yl)ethyl)benzyl)-4-methyl-2...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303980(1-(4-((1H-Tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataKi:  5.06E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303981(Ethyl 3-(4-((4-Methyl-2-propyl-1H-benzo[d]imidazol...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303982(Methyl 3-(4-((4-Methyl-2-propyl-1H-benzo[d]imidazo...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303983(ethyl 2-(4-((4-methyl-2-propyl-1H-benzo[d]imidazol...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303984(Ethyl 2-Methyl-2-(4-((4-methyl-2-propyl-1H-benzo[d...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303985(Ethyl 2,2-Dimethyl-3-(4-(2-(4-methyl-2-propyl-1H-b...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A(Rat)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303986(Ethyl 2-Methyl-3-(4-(2-(4-methyl-2-propyl-1H-benzo...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed