Compile Data Set for Download or QSAR
Report error Found 218 Enz. Inhib. hit(s) with all data for entry = 50031409
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of rat GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash luminescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312779((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312766((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312780((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 4.10nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312776((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312767((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312787(((S)-4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312771((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312799((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 12.2nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312792((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 12.7nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312789((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312786((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 14.3nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312785((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 17.7nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312788((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312781((4-(1H-indole-6-carbonyl)piperazin-1-yl)(3'-methox...)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312777((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312801((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312791((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 33.7nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312790((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 37.2nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312800(((S)-4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312793((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 42.2nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312773((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 46.5nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312769((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312795((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312783((R)-(4-(1H-indole-6-carbonyl)-2-methylpiperazin-1-...)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312774((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312770((4-(1H-indole-6-carbonyl)piperazin-1-yl)(biphenyl-...)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312797((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 123nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312768((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 136nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312794((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 143nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312775((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 147nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312796((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 245nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312782((S)-(4-(1H-indole-6-carbonyl)-2-methylpiperazin-1-...)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312798((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 339nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312772((R)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 640nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312784((4-(1H-indole-6-carbonyl)-1,4-diazepan-1-yl)(biphe...)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312766((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of muscarinic M3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312767((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of muscarinic M3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312768((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of muscarinic M3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312769((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of muscarinic M3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312770((4-(1H-indole-6-carbonyl)piperazin-1-yl)(biphenyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312771((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312772((R)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312773((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312774((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312775((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312776((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
LigandPNGBDBM50312777((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
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