Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50001021
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011972(CHEMBL385189 | Sar-Arg-Val-Tyr-Ile-His-Pro-Thi-OH)
Affinity DataIC50: 0.110nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011977((E)-3-[2-n-butyl-1-{(4-carboxyphenyl)methyl}-1H-im...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011973(CHEMBL216061 | Sar-Arg-Val-Tyr-Ile-His-Pro-Phe | S...)
Affinity DataIC50: 1.30nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011975(4-[2-Butyl-5-(2-carboxy-3-thiophen-2-yl-propenyl)-...)
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011978(CHEMBL40089 | 3-[2-Butyl-3-(4-hydroxy-3-methyl-ben...)
Affinity DataIC50: 21nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011974(CHEMBL291086 | 3-[2-Butyl-3-(2-nitro-benzyl)-3H-im...)
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011971(CHEMBL287936 | 3-[2-Butyl-3-(2-hydroxy-benzyl)-3H-...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003266(CHEMBL289543 | 3-[2-Butyl-3-(2-chloro-benzyl)-3H-i...)
Affinity DataIC50: 440nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011976(CHEMBL287762 | 3-[2-Butyl-3-(4-nitro-benzyl)-3H-im...)
Affinity DataIC50: 620nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003301(CHEMBL36846 | 2-Benzyl-3-[2-butyl-3-(2-chloro-benz...)
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50011970(CHEMBL39349 | 2-[2-Butyl-5-(2-carboxy-3-thiophen-2...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003257(CHEMBL291114 | 3-[2-Butyl-3-(2-chloro-benzyl)-3H-i...)
Affinity DataIC50: 8.90E+3nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003290(CHEMBL39345 | [2-Butyl-3-(2-chloro-benzyl)-3H-imid...)
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003284(CHEMBL25528 | [2-Butyl-5-chloro-3-(2-chloro-benzyl...)
Affinity DataIC50: 4.30E+4nMAssay Description:In vitro inhibition of [125I]AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed