Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50031472
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214864(3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50: 10nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214857(IN-1166 | 3-((5-(6-methylpyridin-2-yl)-4-(quinoxal...)
Affinity DataIC50: 12nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214853(3-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50: 15nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214868(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50: 21nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214866(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50: 24nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214859(4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50: 42nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214861(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50: 46nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214862(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50: 46nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214856(4-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50: 47nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214863(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50: 73nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214865(4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50: 75nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214867(4-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50: 92nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110208(SB-431542 | cid_4521392 | 4-(5-(benzo[d][1,3]dioxo...)
Affinity DataIC50: 94nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214854(3-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50: 119nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214858(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50: 153nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110205(4-(4-Benzo[1,3]dioxol-5-yl-5-pyridin-2-yl-1H-imida...)
Affinity DataIC50: 170nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214860(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50: 171nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110202((4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-...)
Affinity DataIC50: 260nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214869(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50: 262nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214855(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50: 360nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214852(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50: 385nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110199(4-(4-(4-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol...)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Northeastern Ohio Universities Colleges of Medicine and Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110197(4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1...)
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed