Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50031631
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM14777(CHEMBL779 | (6R,12aR)-6-(1,3-benzodioxol-5-yl)-2-m...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316422(CHEMBL1098905 | CHEMBL1099245 | (5R,11aR)-5-(2-Bro...)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316440((6R,12aS)-2-Benzyl-6-(2-bromophenyl)-2,3,6,7,12,12...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316436((6R,12aS)-6-(2-Bromophenyl)-2-ethyl-2,3,6,7,12,12a...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316438((6R,12aS)-6-(2-Bromophenyl)-2-butyl-2,3,6,7,12,12a...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316432((6R,12aS)-6-(2-Bromophenyl)-2-methyl-2,3,6,7,12,12...)
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316429((6R,12aR)-6-(2-Bromophenyl)-2-methyl-2,3,6,7,12,12...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316437((6R,12aR)-6-(2-Bromophenyl)-2-butyl-2,3,6,7,12,12a...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316422(CHEMBL1098905 | CHEMBL1099245 | (5R,11aR)-5-(2-Bro...)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316433((6R,12aR)-6-(2-Bromophenyl)-2-ethyl-2,3,6,7,12,12a...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316423(CHEMBL1099243 | CHEMBL1099244 | (5S,11aR)-5-(2-Bro...)
Affinity DataIC50: 640nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316431((6S,12aS)-6-(2-Bromophenyl)-2-methyl-2,3,6,7,12,12...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316421((1R,3S)Methyl 1-(2-bromophenyl)-2,3,4,9-tetrahydro...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316439((6R,12aR)-2-Benzyl-6-(2-bromophenyl)-2,3,6,7,12,12...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316423(CHEMBL1099243 | CHEMBL1099244 | (5S,11aR)-5-(2-Bro...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316420((1R,3R)Methyl 1-(2-bromophenyl)-2,3,4,9-tetrahydro...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316427((5R-11aS)-5-(2-Bromophenyl)-2-ethyl-1-oxo-5,6,11,1...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316428(Methyl(1R,3R)-1-(2-bromophenyl)-2-(2-chloroacetyl)...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316435((6S,12aS)-6-(2-Bromophenyl)-2-ethyl-2,3,6,7,12,12a...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316434((6S,12aR)-6-(2-Bromophenyl)-2-ethyl-2,3,6,7,12,12a...)
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316426((5S,11aR)-5-(2-Bromophenyl)-2-ethyl-1-oxo-5,6,11,1...)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50316430((6S,12aR)-6-(2-Bromophenyl)-2-methyl-2,3,6,7,12,12...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of human recombinant PDE5 after 1.5 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed