Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50031582
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315759(N-[2-(Dimethylamino)ethyl]-4-[({4-[4-morpholin-4-y...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315762(N-[2-(Dimethylamino)ethyl]-4-({[4-(7-ethyl-4-morph...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315758(N-[2-(Dimethylamino)ethyl]-N-methyl-4-[({4-[4-morp...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315754(1-[4-(7-Ethyl-4-morpholin-4-yl-7H-pyrrolo[2,3-d]py...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315754(1-[4-(7-Ethyl-4-morpholin-4-yl-7H-pyrrolo[2,3-d]py...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315758(N-[2-(Dimethylamino)ethyl]-N-methyl-4-[({4-[4-morp...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315746(1-[4-(4-Morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315747(1-{4-[4-Morpholin-4-yl-7-(2,2,2-trifluoroethyl)-7H...)
Affinity DataIC50: 1nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315748(1-{4-[7-(2,2-Dimethoxyethyl)-4-morpholin-4-yl-7H-p...)
Affinity DataIC50: 1nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315759(N-[2-(Dimethylamino)ethyl]-4-[({4-[4-morpholin-4-y...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315753(1-[4-(7-Ethyl-4-morpholin-4-yl-7H-pyrrolo[2,3-d]py...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315760(1-{4-[(4-Methylpiperazin-1-yl)carbonyl]phenyl}-3-{...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315761(1-(4-{[4-(Dimethylamino)piperidin-1-yl]carbonyl}ph...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315762(N-[2-(Dimethylamino)ethyl]-4-({[4-(7-ethyl-4-morph...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315742(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315757(1-{4-[7-(2-Hydroxyethyl)-4-morpholin-4-yl-7H-pyrro...)
Affinity DataIC50: 2nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315749(1-{4-[4-Morpholin-4-yl-7-(2-oxoethyl)-7H-pyrrolo[2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315760(1-{4-[(4-Methylpiperazin-1-yl)carbonyl]phenyl}-3-{...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315753(1-[4-(7-Ethyl-4-morpholin-4-yl-7H-pyrrolo[2,3-d]py...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315741(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315749(1-{4-[4-Morpholin-4-yl-7-(2-oxoethyl)-7H-pyrrolo[2...)
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315757(1-{4-[7-(2-Hydroxyethyl)-4-morpholin-4-yl-7H-pyrro...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315761(1-(4-{[4-(Dimethylamino)piperidin-1-yl]carbonyl}ph...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315750(1-{4-[4-Morpholin-4-yl-7-(2-pyrrolidin-1-ylethyl)-...)
Affinity DataIC50: 7nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315756(1-{4-[4-Morpholin-4-yl-7-(2-piperazin-1-ylethyl)-7...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315740(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 7nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315742(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315743(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315747(1-{4-[4-Morpholin-4-yl-7-(2,2,2-trifluoroethyl)-7H...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315752(1-{4-[7-(2-{[2-(Dimethylamino)ethyl]amino}ethyl)-4...)
Affinity DataIC50: 11nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315756(1-{4-[4-Morpholin-4-yl-7-(2-piperazin-1-ylethyl)-7...)
Affinity DataIC50: 14nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315741(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315748(1-{4-[7-(2,2-Dimethoxyethyl)-4-morpholin-4-yl-7H-p...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315729(3-{7-[(Dimethylamino)methyl]-4-morpholin-4-yl-5H-p...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315730({3-[4-Morpholin-4-yl-7-(pyrrolidin-1-ylmethyl)-5H-...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315755(1-(4-{7-[2-(4-Methylpiperazin-1-yl)ethyl]-4-morpho...)
Affinity DataIC50: 24nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315743(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315746(1-[4-(4-Morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315750(1-{4-[4-Morpholin-4-yl-7-(2-pyrrolidin-1-ylethyl)-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315744(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315745(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 33nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315752(1-{4-[7-(2-{[2-(Dimethylamino)ethyl]amino}ethyl)-4...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315738((3-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-7H...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315755(1-(4-{7-[2-(4-Methylpiperazin-1-yl)ethyl]-4-morpho...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315737(3-(4-Morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-2-y...)
Affinity DataIC50: 43nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315751(1-{4-[4-Morpholin-4-yl-7-(2-piperidin-1-ylethyl)-7...)
Affinity DataIC50: 52nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315751(1-{4-[4-Morpholin-4-yl-7-(2-piperidin-1-ylethyl)-7...)
Affinity DataIC50: 53nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50315745(1-(4-{7-[2-(Dimethylamino)ethyl]-4-morpholin-4-yl-...)
Affinity DataIC50: 54nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
LigandPNGBDBM50305306((3-(9-(1-benzylpiperidin-4-yl)-6-morpholino-9H-pur...)
Affinity DataIC50: 63nMAssay Description:Inhibition of human PI3Kalpha by fluorescence polarization format assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315737(3-(4-Morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-2-y...)
Affinity DataIC50: 64nMAssay Description:Inhibition of mTOR by DELFIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
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