Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50031602
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50316021((S)-N-((6S,9S,12S,15S,18S)-1-amino-18-carbamoyl-12...)
Affinity DataIC50: 400nMAssay Description:Inhibition of PKB by radioactive kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50316022((S)-N-((6S,9S,12S,15S,18S)-1-amino-15-(aminomethyl...)
Affinity DataIC50: 840nMAssay Description:Inhibition of PKB by radioactive kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50316025((S)-N-((6S,9S,12S,15S,18S)-1-amino-15-(aminomethyl...)
Affinity DataIC50: 920nMAssay Description:Inhibition of PKB by radioactive kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50316026((S)-N-((6S,9S,12S,15S,18S)-1-amino-15-(aminomethyl...)
Affinity DataIC50: 940nMAssay Description:Inhibition of PKB by radioactive kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50316023((S)-1-((S)-2-((S)-2-acetamido-5-guanidinopentanami...)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of PKB by radioactive kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50316024((2S)-2-[(2S)-3-amino-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2...)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of PKB by radioactive kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed