Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 5780
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93394(PSTQ Analog, 3{1,27})
Affinity DataKi:  2.86nM IC50: 6.17nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93364(PSTQ Analog, 3{1,22})
Affinity DataKi:  3.54nM IC50: 7.62nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93393(PSTQ Analog, 3{1,26})
Affinity DataKi:  5.01nM IC50: 10.8nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93392(PSTQ Analog, 3{1,4})
Affinity DataKi:  7.04nM IC50: 15.2nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93385(PSTQ Analog, 3{1,43})
Affinity DataKi:  7.65nM IC50: 16.5nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93376(PSTQ Analog, 3{1,25})
Affinity DataKi:  12.9nM IC50: 27.8nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93363(PSTQ Analog, 3{1,21})
Affinity DataKi:  13.2nM IC50: 28.4nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93400(PSTQ Analog, 3{8,4})
Affinity DataKi:  16.7nM IC50: 35.9nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93399(PSTQ Analog, 3{1,49})
Affinity DataKi:  19.5nM IC50: 42.1nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93395(PSTQ Analog, 3{1,28})
Affinity DataKi:  27.6nM IC50: 59.5nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93397(PSTQ Analog, 3{1,42})
Affinity DataIC50: 30nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93396(PSTQ Analog, 3{1,40})
Affinity DataIC50: 30nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93391(PSTQ Analog, 3{1,3})
Affinity DataKi:  49.5nM IC50: 107nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93363(PSTQ Analog, 3{1,21})
Affinity DataIC50: 75.4nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93362(PSTQ Analog, 3{1,13})
Affinity DataIC50: 128nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93364(PSTQ Analog, 3{1,22})
Affinity DataIC50: 142nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93386(PSTQ Analog, 3{1,44})
Affinity DataIC50: 164nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93382(PSTQ Analog, 3{9,31})
Affinity DataIC50: 295nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93390(PSTQ Analog, 3{1,2})
Affinity DataIC50: 300nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93366(PSTQ Analog, 3{2,12})
Affinity DataIC50: 320nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93372(PSTQ Analog, 3{9,20})
Affinity DataIC50: 356nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93361(PSTQ Analog, 3{1,12})
Affinity DataIC50: 381nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93367(PSTQ Analog, 3{2,13})
Affinity DataIC50: 528nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93385(PSTQ Analog, 3{1,43})
Affinity DataIC50: 564nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93377(PSTQ Analog, 3{3,27})
Affinity DataIC50: 572nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93376(PSTQ Analog, 3{1,25})
Affinity DataIC50: 580nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93371(PSTQ Analog, 3{9,13})
Affinity DataIC50: 603nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93357(PSTQ Analog, 3{2,10})
Affinity DataIC50: 606nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93370(PSTQ Analog, 3{6,20})
Affinity DataIC50: 628nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93384(PSTQ Analog, 3{10,33})
Affinity DataIC50: 670nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93380(PSTQ Analog, 3{7,37})
Affinity DataIC50: 704nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93368(PSTQ Analog, 3{2,20})
Affinity DataIC50: 740nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93381(PSTQ Analog, 3{8,31})
Affinity DataIC50: 770nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93373(PSTQ Analog, 3{9,21})
Affinity DataIC50: 779nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93360(PSTQ Analog, 3{10,4})
Affinity DataIC50: 964nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93387(PSTQ Analog, 3{9,44})
Affinity DataIC50: 971nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93365(PSTQ Analog, 3{1,23})
Affinity DataIC50: 983nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93383(PSTQ Analog, 3{10,32})
Affinity DataIC50: 1.00E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93355(PSTQ Analog, 9)
Affinity DataIC50: 1.05E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93389(PSTQ Analog, 3{9,58})
Affinity DataIC50: 1.20E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93388(PSTQ Analog, 3{9,53})
Affinity DataIC50: 1.31E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93356(PSTQ Analog, 10)
Affinity DataIC50: 1.37E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93379(PSTQ Analog, 3{7,31})
Affinity DataIC50: 1.43E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93374(PSTQ Analog, 3{10,21})
Affinity DataIC50: 1.46E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93369(PSTQ Analog, 3{2,21})
Affinity DataIC50: 1.48E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93375(PSTQ Analog, 3{12,21})
Affinity DataIC50: 1.80E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93358(PSTQ Analog, 3{9,9})
Affinity DataIC50: 2.01E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93359(PSTQ Analog, 3{10,3})
Affinity DataIC50: 2.18E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Chemical Diversity Research Institute

LigandPNGBDBM93354(PSTQ Analog, 8)
Affinity DataIC50: 5.74E+3nMAssay Description:Radioligand binding assay using 5-HT6R.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2013
Entry Details Article
PubMed