Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50031682
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317154(4-[4-(3-Methoxy-phenyl)-2-oxo-2lambda*5*-[1,3,2]di...)
Affinity DataIC50: 270nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317154(4-[4-(3-Methoxy-phenyl)-2-oxo-2lambda*5*-[1,3,2]di...)
Affinity DataIC50: 300nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317152((2R,4S)-4-[4-(3-Chloro-phenyl)-2-oxo-2lambda*5*-[1...)
Affinity DataIC50: 420nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317151((2S,2'S)-diethyl 2,2'-(((6,7-dimethyl-8H-indeno[1,...)
Affinity DataIC50: 580nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317153(4-[4-(4-Chloro-phenyl)-2-oxo-2lambda*5*-[1,3,2]dio...)
Affinity DataIC50: 650nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317153(4-[4-(4-Chloro-phenyl)-2-oxo-2lambda*5*-[1,3,2]dio...)
Affinity DataIC50: 730nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317157(6,7-Dimethyl-4-(2-oxo-4-pyridin-4-yl-2lambda*5*-[1...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317152((2R,4S)-4-[4-(3-Chloro-phenyl)-2-oxo-2lambda*5*-[1...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317156(6,7-Dimethyl-4-(2-oxo-4-pyridin-3-yl-2lambda*5*-[1...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317159(6,7-Dimethyl-4-[4-(6-methyl-pyridin-3-yl)-2-oxo-2l...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317158(6,7-Dimethyl-4-[4-(2-methyl-pyridin-3-yl)-2-oxo-2l...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317155(6,7-Dimethyl-4-(2-oxo-4-pyridin-2-yl-2lambda*5*-[1...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50317160((2R,4S)-6,7-Dimethyl-4-[4-(2-methyl-pyridin-3-yl)-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed