Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50031694
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317420(1-Dehydro-10-gingerdione | CHEMBL1094100)
Affinity DataKi:  3.59E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317425(10-Gingerol | CHEMBL549472)
Affinity DataKi:  3.74E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317423(10-Shogaol | (E)-1-(4-Hydroxy-3-methoxy-phenyl)-te...)
Affinity DataKi:  5.84E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317422(1-Dehydro-6-gingerdione | CHEMBL1096043)
Affinity DataKi:  6.53E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317421(1-Dehydro-8-gingerdione | CHEMBL1096044)
Affinity DataKi:  6.54E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317419(6-Dihydroparadol | CHEMBL1094101)
Affinity DataKi:  9.53E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317426(8-Gingerol | CHEMBL1095671)
Affinity DataKi:  1.17E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50317424(8-Shogaol | (E)-1-(4-Hydroxy-3-methoxy-phenyl)-dod...)
Affinity DataKi:  1.31E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50240419((E)-1-(4-Hydroxy-3-methoxy-phenyl)-dec-4-en-3-one ...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Department of Chemistry and Applied Biosciences

Curated by ChEMBL
LigandPNGBDBM50275147([6]-gingerol | Gingerol | BDBM50317427 | CHEMBL446...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed