Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 5663
Target3-phosphoinositide-dependent protein kinase 1(Human)
Merck Research Laboratories

LigandPNGBDBM92490(Compound # 1)
Affinity DataIC50: 11nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM92490(Compound # 1)
Affinity DataIC50: 14nMAssay Description:384-Well TR-Fret assay using AKT-tide peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Merck Research Laboratories

LigandPNGBDBM26198(Jak Inhibitor 1 | CHEMBL21156 | Compound # 2 | 4-t...)
Affinity DataIC50: 20nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM26198(Jak Inhibitor 1 | CHEMBL21156 | Compound # 2 | 4-t...)
Affinity DataIC50: 28nMAssay Description:384-Well TR-Fret assay using AKT-tide peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Merck Research Laboratories

LigandPNGBDBM92492(Alkaloid 1)
Affinity DataIC50: 5.70E+3nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Merck Research Laboratories

LigandPNGBDBM92493(Alkaloid 2)
Affinity DataIC50: 1.80E+4nMAssay Description:1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM92493(Alkaloid 2)
Affinity DataIC50: 3.00E+4nMAssay Description:384-Well TR-Fret assay using AKT-tide peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM92492(Alkaloid 1)
Affinity DataIC50: 3.00E+4nMAssay Description:384-Well TR-Fret assay using AKT-tide peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed