Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50031791
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319324(1-(3,4-dimethoxyphenyl)-2-(1-m-tolyl-1H-tetrazol-5...)
Affinity DataIC50: 93nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319333(3-(1-(3-chlorophenyl)-1H-tetrazol-5-yl)-1-phenylpr...)
Affinity DataIC50: 114nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319316(1-(3,4-dimethoxyphenyl)-2-(1-phenyl-1H-tetrazol-5-...)
Affinity DataIC50: 116nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319331(2-(1-cyclohexyl-1H-tetrazol-5-ylthio)-1-(3,4-dimet...)
Affinity DataIC50: 183nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319360(1-(3-methoxyphenyl)-3-(1-phenyl-1H-tetrazol-5-yl)p...)
Affinity DataIC50: 215nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319310(3,3-dimethyl-1-(1-phenyl-1H-tetrazol-5-ylthio)buta...)
Affinity DataIC50: 252nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319311(1-phenyl-2-(1-phenyl-1H-tetrazol-5-ylthio)ethanone...)
Affinity DataIC50: 257nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319317(1-phenyl-3-(1-phenyl-1H-tetrazol-5-ylthio)propan-2...)
Affinity DataIC50: 289nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319343(3-(1-(3-methoxyphenyl)-1H-tetrazol-5-yl)-1-phenylp...)
Affinity DataIC50: 304nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319358(1-(3-chlorophenyl)-3-(1-phenyl-1H-tetrazol-5-yl)pr...)
Affinity DataIC50: 310nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319341(1-phenyl-3-(1-phenyl-1H-tetrazol-5-yl)propan-1-one...)
Affinity DataIC50: 359nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319344(3-(1-(4-methoxyphenyl)-1H-tetrazol-5-yl)-1-phenylp...)
Affinity DataIC50: 426nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319318(1-(furan-2-yl)-2-(1-phenyl-1H-tetrazol-5-ylthio)et...)
Affinity DataIC50: 485nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319365(3-(5-(4-methoxyphenyl)-1H-tetrazol-1-yl)-1-phenylp...)
Affinity DataIC50: 493nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319362(1-cyclohexyl-3-(1-phenyl-1H-tetrazol-5-yl)propan-1...)
Affinity DataIC50: 506nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319359(1-(4-dichlorophenyl)-3-(1-phenyl-1H-tetrazol-5-yl)...)
Affinity DataIC50: 539nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319332(3-(1-(4-chlorophenyl)-1H-tetrazol-5-yl)-1-phenylpr...)
Affinity DataIC50: 575nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319334(1-phenyl-3-(1-p-tolyl-1H-tetrazol-5-yl)propan-1-on...)
Affinity DataIC50: 588nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319356(1-(3-fluorophenyl)-3-(1-phenyl-1H-tetrazol-5-yl)pr...)
Affinity DataIC50: 597nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319336(1-phenyl-3-(1-o-tolyl-1H-tetrazol-5-yl)propan-1-on...)
Affinity DataIC50: 683nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319345(4-(5-(3-oxo-3-phenylpropyl)-1H-tetrazol-1-yl)benzo...)
Affinity DataIC50: 686nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319366(3-(5-(benzo[d][1,3]dioxol-5-yl)-1H-tetrazol-1-yl)-...)
Affinity DataIC50: 722nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319364(3-(5-(2-methoxyphenyl)-1H-tetrazol-1-yl)-1-phenylp...)
Affinity DataIC50: 751nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319354(1-phenyl-4-(1-phenyl-1H-tetrazol-5-yl)butan-2-one ...)
Affinity DataIC50: 820nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319363(1-phenyl-3-(5-phenyl-1H-tetrazol-1-yl)propan-1-one...)
Affinity DataIC50: 843nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319329(2-(1-benzyl-1H-tetrazol-5-ylthio)-1-(3,4-dimethoxy...)
Affinity DataIC50: 860nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319351(3-(1-cyclohexyl-1H-tetrazol-5-yl)-1-phenylpropan-1...)
Affinity DataIC50: 915nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319339(3,3-dimethyl-1-(1-phenyl-1H-tetrazol-5-ylsulfonyl)...)
Affinity DataIC50: 943nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319335(1-phenyl-3-(1-m-tolyl-1H-tetrazol-5-yl)propan-1-on...)
Affinity DataIC50: 948nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319321(1-(3,4-dimethoxyphenyl)-2-(1-isopropyl-1H-tetrazol...)
Affinity DataIC50: 954nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319340(1-phenyl-2-(1-phenyl-1H-tetrazol-5-yloxy)ethanone ...)
Affinity DataIC50: 971nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319355(1-phenyl-5-(1-phenyl-1H-tetrazol-5-yl)pentan-3-one...)
Affinity DataIC50: 987nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319350(3-(1-cyclopentyl-1H-tetrazol-5-yl)-1-phenylpropan-...)
Affinity DataIC50: 987nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319326(1-(3,4-dimethoxyphenyl)-2-(1-(2,4-dimethylphenyl)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319328(2-(1-(4-chlorophenyl)-1H-tetrazol-5-ylthio)-1-(3,4...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319314(1-(4-methoxyphenyl)-2-(1-phenyl-1H-tetrazol-5-ylth...)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319368(3-(5-(3-chlorophenyl)-1H-tetrazol-1-yl)-1-phenylpr...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319373(1-phenyl-3-(5-(thiophen-3-yl)-1H-tetrazol-1-yl)pro...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319348(1-phenyl-3-(1-(1,2,3,4-tetrahydronaphthalen-1-yl)-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319338(3,3-dimethyl-1-(1-phenyl-1H-tetrazol-5-ylsulfinyl)...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319312(1-(4-fluorophenyl)-2-(1-phenyl-1H-tetrazol-5-ylthi...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319313(1-(3-fluorophenyl)-2-(1-phenyl-1H-tetrazol-5-ylthi...)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319323(1-(3,4-dimethoxyphenyl)-2-(1-o-tolyl-1H-tetrazol-5...)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319347(3-(1-(2,3-dihydro-1H-inden-1-yl)-1H-tetrazol-5-yl)...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319352(3-[1-(1-adamantyl)-1H-tetrazol-5-yl]-1-phenylpropa...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319315(1-(3-methoxyphenyl)-2-(1-phenyl-1H-tetrazol-5-ylth...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319327(1-(3,4-dimethoxyphenyl)-2-(1-(2-methoxyphenyl)-1H-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319322(2-(1-tert-butyl-1H-tetrazol-5-ylthio)-1-(3,4-dimet...)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319330(1-(3,4-dimethoxyphenyl)-2-(1-(thiophen-2-ylmethyl)...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50319319(2-(1-phenyl-1H-tetrazol-5-ylthio)-1-(thiophen-2-yl...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Displayed 1 to 50 (of 65 total ) | Next | Last >>
Jump to: