Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50004362
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50482166(3-Iodocytisine | CHEMBL187394)
Affinity DataIC50: 0.245nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50329578((-)-9-Bromocytisine | (1R,5S)-9-Bromo-1,2,3,4,5,6-...)
Affinity DataIC50: 0.309nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50143282((1R,9R)-7,11-diazatricyclo[7.3.1.0~2,7~]trideca-2,...)
Affinity DataIC50: 69nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50482165(CHEMBL1083905)
Affinity DataIC50: 102nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50482164(N-Methylcytisine | CHEMBL1085045)
Affinity DataIC50: 112nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50482168(3,5-Dibromocytisine | CHEMBL1084011)
Affinity DataIC50: 372nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Instituto De Investigaciones Biol£Gicas Clemente Estable

Curated by ChEMBL
LigandPNGBDBM50482167(5-Bromocytisine | CHEMBL1084012)
Affinity DataIC50: 457nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed