Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50031841
TargetExportin-1(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50240512(osthole | 7-Methoxy-8-(3-methyl-but-2-enyl)-chrome...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CRM1-mediated hemagglutininin-tagged HIV1 Rev protein nuclear export in human HeLa cells assessed as nucleus localization after 12 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetExportin-1(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50320332(8-(3-methylbut-2-enyl)-2H-chromen-2-one | CHEMBL10...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of CRM1-mediated hemagglutininin-tagged HIV1 Rev protein nuclear export in human HeLa cells assessed as nucleus localization after 12 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetExportin-1(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM12342(2H-chromen-2-one | CHEMBL6466 | Coumarin)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CRM1-mediated hemagglutininin-tagged HIV1 Rev protein nuclear export in human HeLa cells assessed as nucleus localization after 12 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetExportin-1(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50303499(7-(methyloxy)-2H-chromen-2-one | 7-Methoxycoumarin...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CRM1-mediated hemagglutininin-tagged HIV1 Rev protein nuclear export in human HeLa cells assessed as nucleus localization after 12 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetExportin-1(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50320333(7-methoxy-8-(3-methylbut-2-enyl)-2H-chromen-2-one ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CRM1-mediated hemagglutininin-tagged HIV1 Rev protein nuclear export in human HeLa cells assessed as nucleus localization after 12 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed