Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50033623
LigandPNGBDBM50348457(CHEMBL1801207)
Affinity DataIC50: 1nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348465(CHEMBL1801177)
Affinity DataIC50: 2nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348456(CHEMBL1801206)
Affinity DataIC50: 2nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348474(CHEMBL1801186)
Affinity DataIC50: 3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348473(CHEMBL1801185)
Affinity DataIC50: 3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348466(CHEMBL1801178)
Affinity DataIC50: 5nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348468(CHEMBL1801180)
Affinity DataIC50: 5nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348467(CHEMBL1801179)
Affinity DataIC50: 6nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348478(CHEMBL1801205)
Affinity DataIC50: 7nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348454(CHEMBL1801191)
Affinity DataIC50: 8nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348455(CHEMBL1801192)
Affinity DataIC50: 8nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348465(CHEMBL1801177)
Affinity DataIC50: 10nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348470(CHEMBL1801182)
Affinity DataIC50: 20nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348456(CHEMBL1801206)
Affinity DataIC50: 22nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348458(CHEMBL1801208)
Affinity DataIC50: 22nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348460(CHEMBL1801210)
Affinity DataIC50: 22nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348475(CHEMBL1801187)
Affinity DataIC50: 25nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348472(CHEMBL1801184)
Affinity DataIC50: 25nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348464(CHEMBL1801176)
Affinity DataIC50: 32nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348453(CHEMBL1801188)
Affinity DataIC50: 32nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348471(CHEMBL1801183)
Affinity DataIC50: 32nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348459(CHEMBL1801209)
Affinity DataIC50: 42nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348463(CHEMBL1801213)
Affinity DataIC50: 58nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348457(CHEMBL1801207)
Affinity DataIC50: 59nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348469(CHEMBL1801181)
Affinity DataIC50: 79nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348467(CHEMBL1801179)
Affinity DataIC50: 79nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348474(CHEMBL1801186)
Affinity DataIC50: 85nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348468(CHEMBL1801180)
Affinity DataIC50: 126nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348476(CHEMBL1801189)
Affinity DataIC50: 126nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348478(CHEMBL1801205)
Affinity DataIC50: 158nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348462(CHEMBL1801212)
Affinity DataIC50: 169nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348477(CHEMBL1801190)
Affinity DataIC50: 200nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348455(CHEMBL1801192)
Affinity DataIC50: 200nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348461(CHEMBL1801211)
Affinity DataIC50: 213nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50348453(CHEMBL1801188)
Affinity DataIC50: 316nMAssay Description:Inhibition of human hERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348471(CHEMBL1801183)
Affinity DataIC50: 316nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348470(CHEMBL1801182)
Affinity DataIC50: 398nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348464(CHEMBL1801176)
Affinity DataIC50: 398nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348458(CHEMBL1801208)
Affinity DataIC50: 537nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348453(CHEMBL1801188)
Affinity DataIC50: 631nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348472(CHEMBL1801184)
Affinity DataIC50: 631nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348475(CHEMBL1801187)
Affinity DataIC50: 794nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348473(CHEMBL1801185)
Affinity DataIC50: 794nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348459(CHEMBL1801209)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348461(CHEMBL1801211)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348463(CHEMBL1801213)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348462(CHEMBL1801212)
Affinity DataIC50: 1.07E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348466(CHEMBL1801178)
Affinity DataIC50: 1.59E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348476(CHEMBL1801189)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50348469(CHEMBL1801181)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity at voltage-gated calcium channel subunit alpha2delta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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