Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50031999
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50322999(4-(ethoxymethylene)isoquinoline-1,3(2H,4H)-dione |...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50322995(cid_349435 | CHEMBL1210769 | isoquinoline-1,3(2H,4...)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50322996(2,7-naphthyridine-1,3,6,8-tetrone | CHEMBL1210770)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50322997(1,2-dihydroisoquinolin-3(4H)-one | CHEMBL1210771)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50322998(4-(thiophen-2-ylmethylene)isoquinoline-1,3(2H,4H)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50323000(5,7-dichloroquinazoline-2,4(1H,3H)-dione | CHEMBL1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 14(Human)
University of Namur

Curated by ChEMBL
LigandPNGBDBM50012070(CHEMBL295316 | plumbagin | 5-hydroxy-2-methylnapht...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GST-fused NIK expressed in Sf9 cells after 60 mins by radiometric protein kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed