Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50033627
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348617(CHEMBL1801361)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348615(CHEMBL1801359)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348616(CHEMBL1801360)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348614(CHEMBL1801358)
Affinity DataIC50: 82nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348612(CHEMBL1801337)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348611(CHEMBL1801336)
Affinity DataIC50: 92nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348591(CHEMBL1801272)
Affinity DataIC50: 92nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348610(CHEMBL1801335)
Affinity DataIC50: 95nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348608(CHEMBL1801332)
Affinity DataIC50: 96nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348606(CHEMBL1801330)
Affinity DataIC50: 114nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348619(CHEMBL1801333)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348607(CHEMBL1801331)
Affinity DataIC50: 131nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348603(CHEMBL1801327)
Affinity DataIC50: 134nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348609(CHEMBL1801334)
Affinity DataIC50: 138nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348605(CHEMBL1801329)
Affinity DataIC50: 145nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348592(CHEMBL1801317)
Affinity DataIC50: 154nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348613(CHEMBL1801338)
Affinity DataIC50: 239nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348589(CHEMBL1801270)
Affinity DataIC50: 254nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348590(CHEMBL1801271)
Affinity DataIC50: 321nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348593(CHEMBL1801318)
Affinity DataIC50: 336nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348588(CHEMBL1801269)
Affinity DataIC50: 351nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348594(CHEMBL1801319)
Affinity DataIC50: 358nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348587(CHEMBL1801268)
Affinity DataIC50: 369nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348586(CHEMBL1801267)
Affinity DataIC50: 380nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348586(CHEMBL1801267)
Affinity DataIC50: 380nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348596(CHEMBL1801321)
Affinity DataIC50: 387nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348601(CHEMBL1801326)
Affinity DataIC50: 635nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348602(CHEMBL1800088)
Affinity DataIC50: 660nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348604(CHEMBL1801328)
Affinity DataIC50: 851nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348595(CHEMBL1801320)
Affinity DataIC50: 1.33E+3nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348618(CHEMBL1801362)
Affinity DataIC50: 1.46E+3nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348599(CHEMBL1801324)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348597(CHEMBL1801322)
Affinity DataIC50: 1.73E+3nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348600(CHEMBL1801325)
Affinity DataIC50: 2.18E+3nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348598(CHEMBL1801323)
Affinity DataIC50: 3.17E+3nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348617(CHEMBL1801361)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50348614(CHEMBL1801358)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of thromboxane A2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed