Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50035961
TargetGlucocorticoid receptor(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50012202(CHEMBL300409 | 17-(2-Bromo-acetyl)-9-fluoro-11,17-...)
Affinity DataEC50:  8.30E+9nMAssay Description:Partial agonist (20%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50012201(CHEMBL48439 | 9-Fluoro-11,17-dihydroxy-17-[2-(2-is...)
Affinity DataEC50:  9.10E+9nMAssay Description:Partial agonist (48%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50012202(CHEMBL300409 | 17-(2-Bromo-acetyl)-9-fluoro-11,17-...)
Affinity DataIC50: 130nMAssay Description:Partial agonist(20%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50012201(CHEMBL48439 | 9-Fluoro-11,17-dihydroxy-17-[2-(2-is...)
Affinity DataIC50: 440nMAssay Description:Partial agonist(48%) effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50012200(CHEMBL52148 | 2,6-Bis-trifluoromethyl-benzoic acid...)
Affinity DataIC50: 770nMAssay Description:Antagonistic effect against glucocorticoid induced transactivation of tyrosine aminotransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed