Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50032072
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323914(Tamoxifen butyl bromide | CHEMBL1213786)
Affinity DataKi:  13.0nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323912(Tamoxifen ethyl bromide | CHEMBL1213784)
Affinity DataKi:  13.7nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323913(Tamoxifen isopropyl bromide | CHEMBL1213785)
Affinity DataKi:  25.4nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataKi:  31.2nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323911(Tamoxifen methyl iodide | CHEMBL1213783)
Affinity DataKi:  46.3nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed