Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50039207
LigandPNGBDBM50321576(1-(4-(3-aminoazetidine-1-carbonyl)-5-(2-fluoro-4-i...)
Affinity DataIC50: 7nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321561(1-acetyl-4-(2-fluoro-4-iodophenylamino)-N-(2-hydro...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321567((S)-5-acetyl-N-(2,3-dihydroxypropoxy)-2-(2-fluoro-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321577((R)-1-(5-(2-fluoro-4-iodophenylamino)-4-(3-hydroxy...)
Affinity DataIC50: 13nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321572((S)-5-acetyl-4-chloro-N-(2,3-dihydroxypropoxy)-2-(...)
Affinity DataIC50: 13nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321564(5-acetyl-2-[(2-fluoro-4-iodophenyl)amino]-N-(2-hyd...)
Affinity DataIC50: 18nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50321570(5-acetyl-4-chloro-2-(2-fluoro-4-iodophenylamino)-N...)
Affinity DataIC50: 18nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321568(5-acetyl-N-(1,3-dihydroxypropan-2-yloxy)-2-(2-fluo...)
Affinity DataIC50: 19nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321574((S)-5-acetyl-N-(2,3-dihydroxypropoxy)-4-fluoro-2-(...)
Affinity DataIC50: 19nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321566((R)-5-acetyl-N-(2,3-dihydroxypropoxy)-2-(2-fluoro-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321562(1-acetyl-4-(2-fluoro-4-iodophenylamino)-N-(2-hydro...)
Affinity DataIC50: 20nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321573((R)-5-acetyl-N-(2,3-dihydroxypropoxy)-4-fluoro-2-(...)
Affinity DataIC50: 29nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321575(1-(5-(2-fluoro-4-iodophenylamino)-4-(3-hydroxyazet...)
Affinity DataIC50: 30nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321571((R)-5-acetyl-4-chloro-N-(2,3-dihydroxypropoxy)-2-(...)
Affinity DataIC50: 32nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321563(5-acetyl-2-(2-fluoro-4-iodophenylamino)-1-methyl-1...)
Affinity DataIC50: 42nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321565(5-acetyl-2-(2-fluoro-4-iodophenylamino)-N-(3-hydro...)
Affinity DataIC50: 46nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321560(1-acetyl-4-(2-fluoro-4-iodophenylamino)-5-methyl-1...)
Affinity DataIC50: 72nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321569(5-acetyl-2-(2-fluoro-4-iodophenylamino)-N-(3-hydro...)
Affinity DataIC50: 90nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
LigandPNGBDBM50321559(1-acetyl-4-(2-fluoro-4-iodophenylamino)-1H-pyrrole...)
Affinity DataIC50: 220nMAssay Description:Inhibition of MEK1 by cascade assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed