Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50039253
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323659(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 1nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323660(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 2nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323662(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 13nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 17nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323668(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 21nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323666(N-(5-tert-butyl-3-cyano-2-methoxyphenyl)-2-(4-(2-m...)
Affinity DataIC50: 22nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323660(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 25nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323650(N-(3-cyano-5-morpholinophenyl)-2-(4-(2-morpholinoe...)
Affinity DataIC50: 28nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323649(N-(3-tert-butyl-5-cyanophenyl)-2-(4-(2-morpholinoe...)
Affinity DataIC50: 33nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323662(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 38nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323654(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 38nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 39nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323651(N-(5-tert-butyl-3-cyano-2-methoxyphenyl)-2-(4-(2-m...)
Affinity DataIC50: 42nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 44nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323661(N-(5-tert-butyl-3-cyano-2-methoxyphenyl)-2-oxo-2-(...)
Affinity DataIC50: 51nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323654(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 59nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323664(N-(5-tert-butyl-3-cyano-2-methoxyphenyl)-2-oxo-2-(...)
Affinity DataIC50: 60nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323653(N-(5-tert-butyl-3-chloro-2-methoxyphenyl)-2-(4-(2-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323655(5-tert-butyl-N-cyclopropyl-2-methoxy-3-(2-(4-(2-mo...)
Affinity DataIC50: 71nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323659(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 72nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323663(N-(5-tert-butyl-3-cyano-2-methoxyphenyl)-2-oxo-2-(...)
Affinity DataIC50: 78nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323658(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 90nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323655(5-tert-butyl-N-cyclopropyl-2-methoxy-3-(2-(4-(2-mo...)
Affinity DataIC50: 140nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323665(N-(5-tert-butyl-3-cyano-2-methoxyphenyl)-2-(4-(6-f...)
Affinity DataIC50: 190nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323658(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 190nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323656((E)-N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido...)
Affinity DataIC50: 200nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323648(N-(3-tert-butylphenyl)-2-(4-(2-morpholinoethoxy)na...)
Affinity DataIC50: 250nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323652(N-(5-tert-butyl-2-methoxyphenyl)-2-(4-(2-morpholin...)
Affinity DataIC50: 250nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323648(N-(3-tert-butylphenyl)-2-(4-(2-morpholinoethoxy)na...)
Affinity DataIC50: 310nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323657(N-(5-tert-butyl-2-methoxy-3-(methylsulfonamido)phe...)
Affinity DataIC50: 390nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
K£Mia

Curated by ChEMBL
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed