Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50039270
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392(SRIF-28 | (4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,3...)
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 9.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 12.3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 16.5nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 29nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 44nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 57.5nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 92.5nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 101nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 161nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 249nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 346nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 356nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 412nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 418nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 892nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed