Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50032199
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325890(N-(1-((6-(benzo[d][1,3]dioxol-4-yl)pyridin-2-yl)me...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325894(N-(3-((6-(benzo[d][1,3]dioxol-4-yl)pyridin-2-yl)me...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325888(N-(1-((6-(benzo[d][1,3]dioxol-4-yl)pyridin-2-yl)me...)
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325892(N-(3-((6-(benzo[d][1,3]dioxol-4-yl)pyridin-2-yl)me...)
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325895(N-(3-((6-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)me...)
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325882(N-(1-((6-(benzo[d][1,3]dioxol-4-yl)pyridin-2-yl)me...)
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325891(N-(1-((6-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)me...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325893(N-(3-((6-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)me...)
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325886(N-(3-(3-(benzo[d][1,3]dioxol-4-yl)benzyl)-1-methyl...)
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325887(N-(3-((4'-fluoro-2'-methoxybiphenyl-3-yl)methyl)-1...)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325889(N-(1-((6-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)me...)
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325884(N-(1-(3-(benzo[d][1,3]dioxol-4-yl)benzyl)-1H-indol...)
Affinity DataIC50: 51nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325885(N-(1-((4'-fluoro-2'-methoxybiphenyl-3-yl)methyl)-1...)
Affinity DataIC50: 58nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325880(N-(1-(3-(benzo[d][1,3]dioxol-4-yl)benzyl)-1H-benzo...)
Affinity DataIC50: 64nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325883(N-(1-((6-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)me...)
Affinity DataIC50: 73nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325879(N-(3-fluorobenzyl)-1-((2'-methoxybiphenyl-3-yl)met...)
Affinity DataIC50: 104nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325881(N-(1-((4'-fluoro-2'-methoxybiphenyl-3-yl)methyl)-1...)
Affinity DataIC50: 269nMAssay Description:Displacement of [3H]CC55940 human cannabinoid CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed