Compile Data Set for Download or QSAR
Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 50041866
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417349(CHEMBL1276248)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-2-imidazoline | 2-(2,6-dic...)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417351(CHEMBL1278084)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412260(CHEMBL273485)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417351(CHEMBL1278084)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417351(CHEMBL1278084)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417349(CHEMBL1276248)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataEC50:  47nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-2-imidazoline | 2-(2,6-dic...)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417349(CHEMBL1276248)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417346(CHEMBL1276220)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417343(CHEMBL1276140)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417341(CHEMBL397753)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataEC50:  76nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417352(CHEMBL1278085)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417348(CHEMBL1276247)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417342(CHEMBL1276139)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417353(CHEMBL242265)
Affinity DataEC50:  112nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417352(CHEMBL1278085)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  115nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417349(CHEMBL1276248)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417348(CHEMBL1276247)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412260(CHEMBL273485)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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