Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50041877
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50060964(5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]...)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50060964(5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417541(CHEMBL1630938)
Affinity DataKi:  0.245nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417542(CHEMBL1630939)
Affinity DataKi:  0.324nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417541(CHEMBL1630938)
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417542(CHEMBL1630939)
Affinity DataKi:  0.347nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417540(CHEMBL1630940)
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50060964(5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]...)
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417540(CHEMBL1630940)
Affinity DataKi:  0.955nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417541(CHEMBL1630938)
Affinity DataKi:  1.91nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417542(CHEMBL1630939)
Affinity DataKi:  2.09nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417540(CHEMBL1630940)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417538(CHEMBL1630942)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417538(CHEMBL1630942)
Affinity DataKi:  15.5nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417539(CHEMBL1630941)
Affinity DataKi:  17.4nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417539(CHEMBL1630941)
Affinity DataKi:  19.1nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417538(CHEMBL1630942)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417539(CHEMBL1630941)
Affinity DataKi:  67.6nMAssay Description:Displacement of [3H]prazosin from human Alpha-1B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed