Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50032548
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50330860(Methylergometrine | CHEMBL1201356 | METHYLERGONOVI...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50060417(CHEMBL297784 | SB 206553 | SB-206553 | 5-Methyl-3,...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  33.1nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM85067(CAS_170856-41-4 | PNU 96415E | CHEMBL81330 | PNU-9...)
Affinity DataKi:  69.6nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM26948(CHEMBL46516 | cid_3396 | FLUSPIRILENE | 8-[4,4-bis...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194444(6-methoxy-1-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,...)
Affinity DataKi:  491nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50330861((5-methoxy-1H-indol-3-yl)methanamine | CHEMBL12760...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50330858(6-Fluoromelatonin | N-[2-(6-Fluoro-5-methoxy-1H-in...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM61401(FENDILINE HYDROCHLORIDE | MLS000069570 | CHEMBL254...)
Affinity DataKi:  3.22E+3nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50330859(10-Hydroxy-10,11-dihydro-dibenzo[b,f]azepine-5-car...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed