Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50032668
TargetProstaglandin G/H synthase 1(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human platelets COX1 after 2 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant COX2 after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50332956((2RS,4R)-2-(1-phenyl-3-p-tolyl-1H-pyrazol-4-yl)thi...)
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant COX2 after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50332955((2RS,4R)-2-(1,3-diphenyl-1H-pyrazol-4-yl)thiazolid...)
Affinity DataIC50: 470nMAssay Description:Inhibition of human recombinant COX2 after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50332954((2RS,4R)-2-(1-phenyl-3-p-tolyl-1H-pyrazol-4-yl)thi...)
Affinity DataIC50: 940nMAssay Description:Inhibition of human recombinant COX2 after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of human recombinant COX2 after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 1(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50332954((2RS,4R)-2-(1-phenyl-3-p-tolyl-1H-pyrazol-4-yl)thi...)
Affinity DataIC50: 9.62E+4nMAssay Description:Inhibition of human platelets COX1 after 2 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50332955((2RS,4R)-2-(1,3-diphenyl-1H-pyrazol-4-yl)thiazolid...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelets COX1 after 2 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelets COX1 after 2 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50332956((2RS,4R)-2-(1-phenyl-3-p-tolyl-1H-pyrazol-4-yl)thi...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelets COX1 after 2 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2011
Entry Details Article
PubMed