Compile Data Set for Download or QSAR
Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 50032582
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331461(1-Trifluoromethyl-cyclopropanecarboxylic acid{3-[(...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331462(1-Trifluoromethyl-cyclobutanecarboxylic acid{3-[(6...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331463(2,2-Difluoro-cyclopropanecarboxylic acid{3-[(6-flu...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331464(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331465(Furan-3-carboxylic acid{3-[(6-fluoro-1,1-dioxo-1H-...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331466(N-{3-[(1,1-Dioxo-1H-1lambda*6*-benzo[d]isothiazol-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331467(1-Methyl-cyclopropanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331468(Furan-2-carboxylic acid{3-[(6-fluoro-1,1-dioxo-1H-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331469(N-{3-[(6-Fluoro-1,1-dioxo-1H-1lambda*6*-benzo[d]is...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331470(Pyrazine-2-carboxylic acid{3-[(6-fluoro-1,1-dioxo-...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331461(1-Trifluoromethyl-cyclopropanecarboxylic acid{3-[(...)
Affinity DataIC50: 240nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331471(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331464(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331472(Cyclopropanecarboxylic acid{3-[(6-fluoro-1,1-dioxo...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331473(Thiazole-4-carboxylic acid{3-[(6-fluoro-1,1-dioxo-...)
Affinity DataIC50: 290nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331474(Pyrrole-1-carboxylic acid{3-[(6-fluoro-1,1-dioxo-1...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331462(1-Trifluoromethyl-cyclobutanecarboxylic acid{3-[(6...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331475(3-Hydroxy-pyridine-2-carboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331463(2,2-Difluoro-cyclopropanecarboxylic acid{3-[(6-flu...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331476(4-Cyano-tetrahydro-pyran-4-carboxylic acid{3-[(6-f...)
Affinity DataIC50: 330nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331477(Morpholine-4-carboxylic acid{3-[(6-fluoro-1,1-diox...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331474(Pyrrole-1-carboxylic acid{3-[(6-fluoro-1,1-dioxo-1...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331478(1-Cyano-cyclopropanecarboxylic acid{3-[(6-fluoro-1...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331479(1-Hydroxy-cyclohexanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331470(Pyrazine-2-carboxylic acid{3-[(6-fluoro-1,1-dioxo-...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331480(Tetrahydro-furan-2-carboxylic acid{3-[(6-fluoro-1,...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331465(Furan-3-carboxylic acid{3-[(6-fluoro-1,1-dioxo-1H-...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331467(1-Methyl-cyclopropanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50: 370nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331469(N-{3-[(6-Fluoro-1,1-dioxo-1H-1lambda*6*-benzo[d]is...)
Affinity DataIC50: 370nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331481(4,4-Difluoro-1-hydroxy-cyclohexanecarboxylic acid{...)
Affinity DataIC50: 390nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331468(Furan-2-carboxylic acid{3-[(6-fluoro-1,1-dioxo-1H-...)
Affinity DataIC50: 410nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331482(N-{3-[(1,1-Dioxo-1H-1lambda*6*-benzo[d]isothiazol-...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331483(Tetrahydro-pyran-2-carboxylic acid{3-[(6-fluoro-1,...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331479(1-Hydroxy-cyclohexanecarboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331475(3-Hydroxy-pyridine-2-carboxylic acid{3-[(6-fluoro-...)
Affinity DataIC50: 460nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331484(1-Hydroxy-cyclopentanecarboxylic acid{3-[(6-fluoro...)
Affinity DataIC50: 470nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331485(Morpholine-4-carboxylic acid{3-[(1,1-dioxo-1H-1lam...)
Affinity DataIC50: 470nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331471(3,3,3-Trifluoro-N-{3-[(6-fluoro-1,1-dioxo-1H-1lamb...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331472(Cyclopropanecarboxylic acid{3-[(6-fluoro-1,1-dioxo...)
Affinity DataIC50: 490nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331486(1-Methyl-1H-imidazole-2-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50: 520nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331487(1-Amino-cyclopropanecarboxylic acid{3-[(6-fluoro-1...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331488(Tetrahydro-pyran-4-carboxylic acid{3-[(6-fluoro-1,...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331473(Thiazole-4-carboxylic acid{3-[(6-fluoro-1,1-dioxo-...)
Affinity DataIC50: 540nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331478(1-Cyano-cyclopropanecarboxylic acid{3-[(6-fluoro-1...)
Affinity DataIC50: 540nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331423(N-{3-[(1,1-Dioxo-1H-1lambda*6*-benzo[d]isothiazol-...)
Affinity DataIC50: 550nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331486(1-Methyl-1H-imidazole-2-carboxylic acid{3-[(6-fluo...)
Affinity DataIC50: 550nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331489(N-{3-[(1,1-Dioxo-1H-1lambda*6*-benzo[d]isothiazol-...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331476(4-Cyano-tetrahydro-pyran-4-carboxylic acid{3-[(6-f...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331481(4,4-Difluoro-1-hydroxy-cyclohexanecarboxylic acid{...)
Affinity DataIC50: 630nMAssay Description:Inhibition of human Kv1.5 ion channel expressed in CHO K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331483(Tetrahydro-pyran-2-carboxylic acid{3-[(6-fluoro-1,...)
Affinity DataIC50: 640nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
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