Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 4637
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81438(CDK Inhibitor, 11)
Affinity DataKi:  0.110nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81433(CDK Inhibitor, 6)
Affinity DataKi:  0.290nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81441(CDK Inhibitor, 14)
Affinity DataKi:  0.380nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81439(CDK Inhibitor, 12)
Affinity DataKi:  0.520nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81440(CDK Inhibitor, 13)
Affinity DataKi:  0.560nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81430(CDK Inhibitor, 3)
Affinity DataKi:  0.800nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81434(CDK Inhibitor, 7)
Affinity DataKi:  0.960nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM8061(4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-(3-nitroph...)
Affinity DataKi: <1nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81433(CDK Inhibitor, 6)
Affinity DataKi:  1.60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81439(CDK Inhibitor, 12)
Affinity DataKi:  1.90nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81441(CDK Inhibitor, 14)
Affinity DataKi:  2.30nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81430(CDK Inhibitor, 3)
Affinity DataKi:  2.40nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Cyclacel

LigandPNGBDBM81440(CDK Inhibitor, 13)
Affinity DataKi:  3nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Cyclacel

LigandPNGBDBM81438(CDK Inhibitor, 11)
Affinity DataKi:  4.10nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81431(CDK Inhibitor, 4)
Affinity DataKi:  4.30nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81432(CDK Inhibitor, 5)
Affinity DataKi:  4.30nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81429(CDK Inhibitor, 2)
Affinity DataKi:  4.5nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM8061(4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-(3-nitroph...)
Affinity DataKi:  4.60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81435(CDK Inhibitor, 8)
Affinity DataKi:  5.90nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81440(CDK Inhibitor, 13)
Affinity DataKi:  5.90nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81436(CDK Inhibitor, 9)
Affinity DataKi:  6.70nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81439(CDK Inhibitor, 12)
Affinity DataKi:  6.80nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81434(CDK Inhibitor, 7)
Affinity DataKi:  7.60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81437(CDK Inhibitor, 10)
Affinity DataKi:  8.5nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81430(CDK Inhibitor, 3)
Affinity DataKi:  9.10nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Cyclacel

LigandPNGBDBM81438(CDK Inhibitor, 11)
Affinity DataKi:  14nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM8061(4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-(3-nitroph...)
Affinity DataKi:  19nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81431(CDK Inhibitor, 4)
Affinity DataKi:  20nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81430(CDK Inhibitor, 3)
Affinity DataKi:  25nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81432(CDK Inhibitor, 5)
Affinity DataKi:  26nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81440(CDK Inhibitor, 13)
Affinity DataKi:  28nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81431(CDK Inhibitor, 4)
Affinity DataKi:  33nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81434(CDK Inhibitor, 7)
Affinity DataKi:  47nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81435(CDK Inhibitor, 8)
Affinity DataKi:  47nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81429(CDK Inhibitor, 2)
Affinity DataKi:  56nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81440(CDK Inhibitor, 13)
Affinity DataKi:  60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Cyclacel

LigandPNGBDBM81430(CDK Inhibitor, 3)
Affinity DataKi:  67nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81441(CDK Inhibitor, 14)
Affinity DataKi:  68nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Cyclacel

LigandPNGBDBM8061(4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-(3-nitroph...)
Affinity DataKi:  73nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM8061(4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-(3-nitroph...)
Affinity DataKi:  73nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Cyclacel

LigandPNGBDBM81433(CDK Inhibitor, 6)
Affinity DataKi:  86nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81433(CDK Inhibitor, 6)
Affinity DataKi:  91nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81433(CDK Inhibitor, 6)
Affinity DataKi:  94nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81439(CDK Inhibitor, 12)
Affinity DataKi:  102nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81431(CDK Inhibitor, 4)
Affinity DataKi:  107nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Cyclacel

LigandPNGBDBM81432(CDK Inhibitor, 5)
Affinity DataKi:  127nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81429(CDK Inhibitor, 2)
Affinity DataKi:  132nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81434(CDK Inhibitor, 7)
Affinity DataKi:  139nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Cyclacel

LigandPNGBDBM81441(CDK Inhibitor, 14)
Affinity DataKi:  149nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Cyclacel

LigandPNGBDBM81432(CDK Inhibitor, 5)
Affinity DataKi:  163nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2011
Entry Details Article
PubMed
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