Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50032755
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50081950(6-hydroxy-2-phenyl-4H-chromen-4-one | NSC-26744 | ...)
Affinity DataIC50: 5.17E+3nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM23419(CHEMBL9352 | (2S)-5,7-dihydroxy-2-(4-hydroxyphenyl...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM7461(5,7-dihydroxy-2-phenyl-4H-chromen-4-one | cid_5281...)
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM26664(7-Hydroxy-flavone, 5a | 7-Hydroxyflavone, 11 | 7-h...)
Affinity DataIC50: 3.71E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50187668(3-hydroxy-2-phenyl-4H-chromen-4-one | 3-Hydroxyfla...)
Affinity DataIC50: 5.52E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM61776((2S)-5-hydroxy-2-(3-hydroxy-4-methoxyphenyl)-7-[[(...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of calmodulin assessed as inhibition of calmodulin-calcium-PDE4 complex formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM61776((2S)-5-hydroxy-2-(3-hydroxy-4-methoxyphenyl)-7-[[(...)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of calmodulin assessed as inhibition of calmodulin-calcium-PDE1 complex formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
Universidad Aut£Noma Del Estado De Morelos

Curated by ChEMBL
LigandPNGBDBM50028962(flavone | CHEMBL275638)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed