Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50039379
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336806(1-(3-(aminomethyl)-2-isobutyl-4-p-tolylquinolin-6-...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336820([5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336805(6-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336803(4-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336804(5-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336819([5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4...)
Affinity DataIC50: 10nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-6-isobutyl-2-methyl-4-p-tolylnicot...)
Affinity DataIC50: 18nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50: 19nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808([5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336802(3-[3-(Aminomethyl)-4-(4-methylphenyl)-2-(2-methylp...)
Affinity DataIC50: 23nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50: 39nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336811(5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-prop...)
Affinity DataIC50: 57nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336812(5-(Aminomethyl)-6-butyl-2-methyl-4-(4-methylphenyl...)
Affinity DataIC50: 58nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336810((2E)-3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl...)
Affinity DataIC50: 66nMAssay Description:Inhibition of DPP4 in human Caco2 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 420nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 630nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50: 820nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336815(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336817(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-4-(4-methyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336814(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-(...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-6-isobutyl-2-methyl-4-p-tolylnicot...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336818(5-(Aminomethyl)-2-benzyl-6-(2,2-dimethylpropyl)-4-...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336816(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-(1-methyl...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336812(5-(Aminomethyl)-6-butyl-2-methyl-4-(4-methylphenyl...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-6-isobutyl-2-methyl-4-p-tolylnicot...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336813(5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50333184(5-(aminomethyl)-6-isobutyl-2-methyl-4-p-tolylnicot...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808([5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336809(3-[5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808([5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336808([5-(Aminomethyl)-2-methyl-4-(4-methylphenyl)-6-(2-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of rat kidney DPP2 after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336820([5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of FLAG-tagged human DPP9 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336820([5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-ethyl-4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336819([5-(Aminomethyl)-6-(2,2-dimethylpropyl)-2-methyl-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of FLAG-tagged human DPP8 expressed in human 293F cells after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
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