Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50033279
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342704(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342709(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-3,4...)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM84637(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342710(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,3...)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342713(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342715(3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)p...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in dhfr-deficient CHO cells assessed as [3H]thymidine incorporationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342704(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342706(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342715(3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)p...)
Affinity DataKi:  0.210nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342719(2,4-dimethyl-5-(4-methyl-5-(3-(5-(4-(trifluorometh...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342713(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342710(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,3...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342711(7-methoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342705(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342717(4'-Acetyl-biphenyl-4-carboxylic acid {4-[4-(2-meth...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342708(3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)pip...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50119390(Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dic...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342711(7-methoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)...)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342707(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-o...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342710(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,3...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342712(6-fluoro-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)b...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342709(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-3,4...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342716(N-(4-(2-((3aR,9bS)-8-cyano-1,3a,4,9b-tetrahydrochr...)
Affinity DataKi:  2nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342705(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50177354(A-437203 | 2-(3-(4-(2-tert-butyl-6-(trifluoromethy...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342720((R)-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342711(7-methoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342710(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,3...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342718(4-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(4-(2-(7-(meth...)
Affinity DataKi:  4nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342715(3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)p...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342705(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342704(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342709(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-3,4...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342706(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342708(3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)pip...)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342712(6-fluoro-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)b...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342704(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342714(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342706(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342713(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342715(3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)p...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342709(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-3,4...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342707(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-o...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342708(3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)pip...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342712(6-fluoro-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)b...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342707(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-o...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342713(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342714(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342714(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Pig)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50342706(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
Displayed 1 to 50 (of 73 total ) | Next | Last >>
Jump to: