Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50032910
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataKi:  500nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of aminopeptidase activity of human leukotriene A4 hydrolase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336495(7-Amino-5,7,8,9-tetrahydro-benzocyclohepten-6-one,...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336493(1-Aminoindan-2-one, hydrochloride | CHEMBL1668624)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336499(cis-7-amino-6,7,8,9-tetrahydro-5H-benzocyclohepten...)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336496(2-aminocycloheptanone hydrochloride | CHEMBL166862...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336497(7-Amino-5,7,8,9-tetrahydrobenzocyclohepten-6-one,6...)
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336498(trans-7-amino-6,7,8,9-tetrahydro-5H-benzocyclohept...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336496(2-aminocycloheptanone hydrochloride | CHEMBL166862...)
Affinity DataIC50: 3.10E+5nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of aminopeptidase activity of human leukotriene A4 hydrolase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336494(6-amino-5,6,8,9-tetrahydrobenzocycloheptene-7-one,...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human aminopeptidase N by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336493(1-Aminoindan-2-one, hydrochloride | CHEMBL1668624)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of aminopeptidase activity of human leukotriene A4 hydrolase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336494(6-amino-5,6,8,9-tetrahydrobenzocycloheptene-7-one,...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of aminopeptidase activity of human leukotriene A4 hydrolase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336495(7-Amino-5,7,8,9-tetrahydro-benzocyclohepten-6-one,...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336497(7-Amino-5,7,8,9-tetrahydrobenzocyclohepten-6-one,6...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336499(cis-7-amino-6,7,8,9-tetrahydro-5H-benzocyclohepten...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336493(1-Aminoindan-2-one, hydrochloride | CHEMBL1668624)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336494(6-amino-5,6,8,9-tetrahydrobenzocycloheptene-7-one,...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336495(7-Amino-5,7,8,9-tetrahydro-benzocyclohepten-6-one,...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of aminopeptidase activity of human leukotriene A4 hydrolase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Merck Sharpe and Dohme

Curated by ChEMBL
LigandPNGBDBM50336497(7-Amino-5,7,8,9-tetrahydrobenzocyclohepten-6-one,6...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of aminopeptidase activity of human leukotriene A4 hydrolase by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed